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Metabolomics-assisted discovery of a new anticancer GLS-1 inhibitor chemotype from a nortopsentin-inspired library: From phenotype screening to target identification.
Carbone D, Vestuto V, Ferraro MR, Ciaglia T, Pecoraro C, Sommella E, Cascioferro S, Salviati E, Novi S, Tecce MF, Amodio G, Iraci N, Cirrincione G, Campiglia P, Diana P, Bertamino A, Parrino B, Ostacolo C. Carbone D, et al. Among authors: bertamino a. Eur J Med Chem. 2022 Apr 15;234:114233. doi: 10.1016/j.ejmech.2022.114233. Epub 2022 Mar 6. Eur J Med Chem. 2022. PMID: 35286926
Design, synthesis, and cytotoxic evaluation of a new series of 3-substituted spiro[(dihydropyrazine-2,5-dione)-6,3'-(2',3'-dihydrothieno[2,3-b]naphtho-4',9'-dione)] derivatives.
Gomez-Monterrey I, Campiglia P, Carotenuto A, Califano D, Pisano C, Vesci L, Lama T, Bertamino A, Sala M, di Bosco AM, Grieco P, Novellino E. Gomez-Monterrey I, et al. Among authors: bertamino a. J Med Chem. 2007 Apr 19;50(8):1787-98. doi: 10.1021/jm0612158. Epub 2007 Mar 22. J Med Chem. 2007. PMID: 17375902
Spiro[(dihydropyrazin-2,5-dione)-6,3'-(2',3'-dihydrothieno[2,3-b]naphtho-4',9'-dione)]-based cytotoxic agents: structure-activity relationship studies on the substituent at N4-position of the diketopiperazine domain.
Gomez-Monterrey I, Campiglia P, Carotenuto A, Stiuso P, Bertamino A, Sala M, Aquino C, Grieco P, Morello S, Pinto A, Ianelli P, Novellino E. Gomez-Monterrey I, et al. Among authors: bertamino a. J Med Chem. 2008 May 22;51(10):2924-32. doi: 10.1021/jm7013056. Epub 2008 Apr 23. J Med Chem. 2008. PMID: 18429610
A novel quinone-based derivative (DTNQ-Pro) induces apoptotic death via modulation of heat shock protein expression in Caco-2 cells.
Gomez-Monterrey I, Campiglia P, Bertamino A, Aquino C, Sala M, Grieco P, Dicitore A, Vanacore D, Porta A, Maresca B, Novellino E, Stiuso P. Gomez-Monterrey I, et al. Among authors: bertamino a. Br J Pharmacol. 2010 Jun;160(4):931-40. doi: 10.1111/j.1476-5381.2010.00718.x. Br J Pharmacol. 2010. PMID: 20590589 Free PMC article.
Identification of the spiro(oxindole-3,3'-thiazolidine)-based derivatives as potential p53 activity modulators.
Gomez-Monterrey I, Bertamino A, Porta A, Carotenuto A, Musella S, Aquino C, Granata I, Sala M, Brancaccio D, Picone D, Ercole C, Stiuso P, Campiglia P, Grieco P, Ianelli P, Maresca B, Novellino E. Gomez-Monterrey I, et al. Among authors: bertamino a. J Med Chem. 2010 Dec 9;53(23):8319-29. doi: 10.1021/jm100838z. Epub 2010 Nov 8. J Med Chem. 2010. PMID: 21058726
Design, synthesis, and cytotoxic evaluation of acyl derivatives of 3-aminonaphtho[2,3-b]thiophene-4,9-dione, a quinone-based system.
Gomez-Monterrey I, Campiglia P, Aquino C, Bertamino A, Granata I, Carotenuto A, Brancaccio D, Stiuso P, Scognamiglio I, Rusciano MR, Maione AS, Illario M, Grieco P, Maresca B, Novellino E. Gomez-Monterrey I, et al. Among authors: bertamino a. J Med Chem. 2011 Jun 23;54(12):4077-91. doi: 10.1021/jm200094h. Epub 2011 May 23. J Med Chem. 2011. PMID: 21553829
Characterization of a selective CaMKII peptide inhibitor.
Gomez-Monterrey I, Sala M, Rusciano MR, Monaco S, Maione AS, Iaccarino G, Tortorella P, D'Ursi AM, Scrima M, Carotenuto A, De Rosa G, Bertamino A, Vernieri E, Grieco P, Novellino E, Illario M, Campiglia P. Gomez-Monterrey I, et al. Among authors: bertamino a. Eur J Med Chem. 2013 Apr;62:425-34. doi: 10.1016/j.ejmech.2012.12.053. Epub 2013 Jan 22. Eur J Med Chem. 2013. PMID: 23395965
72 results