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A fluorine scan of a tubulin polymerization inhibitor isocombretastatin A-4: Design, synthesis, molecular modelling, and biological evaluation.
Naret T, Bignon J, Bernadat G, Benchekroun M, Levaique H, Lenoir C, Dubois J, Pruvost A, Saller F, Borgel D, Manoury B, Leblais V, Darrigrand R, Apcher S, Brion JD, Schmitt E, Leroux FR, Alami M, Hamze A. Naret T, et al. Among authors: bernadat g. Eur J Med Chem. 2018 Jan 1;143:473-490. doi: 10.1016/j.ejmech.2017.11.055. Epub 2017 Dec 2. Eur J Med Chem. 2018. PMID: 29202409
Discovery of azaisoerianin derivatives as potential antitumors agents.
Soussi MA, Provot O, Bernadat G, Bignon J, Wdzieczak-Bakala J, Desravines D, Dubois J, Brion JD, Messaoudi S, Alami M. Soussi MA, et al. Among authors: bernadat g. Eur J Med Chem. 2014 May 6;78:178-89. doi: 10.1016/j.ejmech.2014.03.032. Epub 2014 Mar 13. Eur J Med Chem. 2014. PMID: 24681982
Synthesis, biological evaluation, and structure-activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors.
Aziz J, Brachet E, Hamze A, Peyrat JF, Bernadat G, Morvan E, Bignon J, Wdzieczak-Bakala J, Desravines D, Dubois J, Tueni M, Yassine A, Brion JD, Alami M. Aziz J, et al. Among authors: bernadat g. Org Biomol Chem. 2013 Jan 21;11(3):430-42. doi: 10.1039/c2ob26253c. Epub 2012 Oct 9. Org Biomol Chem. 2013. PMID: 23047722
Diversity-oriented synthesis of fused thioglycosyl benzo[e][1,4]oxathiepin-5-ones and benzo[f][1,4]thiazepin-5(2H)-ones by a sequence of palladium-catalyzed glycosyl thiol arylation and deprotection-lactonization reactions.
AL-Shuaeeb RA, Galvani G, Bernadat G, Brion JD, Alami M, Messaoudi S. AL-Shuaeeb RA, et al. Among authors: bernadat g. Org Biomol Chem. 2015 Nov 28;13(44):10904-16. doi: 10.1039/c5ob01603g. Epub 2015 Sep 15. Org Biomol Chem. 2015. PMID: 26369372
Design, Synthesis, and Biological Activity of New N-(Phenylmethyl)-benzoxazol-2-thiones as Macrophage Migration Inhibitory Factor (MIF) Antagonists: Efficacies in Experimental Pulmonary Hypertension.
Le Hiress M, Akagah B, Bernadat G, Tu L, Thuillet R, Huertas A, Phan C, Fadel E, Simonneau G, Humbert M, Jalce G, Guignabert C. Le Hiress M, et al. Among authors: bernadat g. J Med Chem. 2018 Apr 12;61(7):2725-2736. doi: 10.1021/acs.jmedchem.7b01312. Epub 2018 Mar 19. J Med Chem. 2018. PMID: 29526099
45 results