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Biorefining Twin Transition: Digitalisation for Bio-based Chemicals/Materials - Discovery, Design and Optimisation.
Chimia (Aarau). 2023 Dec 20;77(12):816-826. doi: 10.2533/chimia.2023.816.
Chimia (Aarau). 2023.
PMID: 38131404
Free article.
Top Selling (2026) Small Molecule Orphan Drugs: A Journey into Their Chemistry.
Benedetto Tiz D, Bagnoli L, Rosati O, Marini F, Sancineto L, Santi C.
Benedetto Tiz D, et al.
Int J Mol Sci. 2023 Jan 4;24(2):930. doi: 10.3390/ijms24020930.
Int J Mol Sci. 2023.
PMID: 36674441
Free PMC article.
Review.
Item in Clipboard
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa.
Cotman AE, Durcik M, Benedetto Tiz D, Fulgheri F, Secci D, Sterle M, Možina Š, Skok Ž, Zidar N, Zega A, Ilaš J, Peterlin Mašič L, Tomašič T, Hughes D, Huseby DL, Cao S, Garoff L, Berruga Fernández T, Giachou P, Crone L, Simoff I, Svensson R, Birnir B, Korol SV, Jin Z, Vicente F, Ramos MC, de la Cruz M, Glinghammar B, Lenhammar L, Henderson SR, Mundy JEA, Maxwell A, Stevenson CEM, Lawson DM, Janssen GV, Sterk GJ, Kikelj D.
Cotman AE, et al. Among authors: benedetto tiz d.
J Med Chem. 2023 Jan 26;66(2):1380-1425. doi: 10.1021/acs.jmedchem.2c01597. Epub 2023 Jan 12.
J Med Chem. 2023.
PMID: 36634346
Free PMC article.
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FDA-Approved Small Molecules in 2022: Clinical Uses and Their Synthesis.
Benedetto Tiz D, Bagnoli L, Rosati O, Marini F, Santi C, Sancineto L.
Benedetto Tiz D, et al.
Pharmaceutics. 2022 Nov 21;14(11):2538. doi: 10.3390/pharmaceutics14112538.
Pharmaceutics. 2022.
PMID: 36432728
Free PMC article.
Review.
Item in Clipboard
New Halogen-Containing Drugs Approved by FDA in 2021: An Overview on Their Syntheses and Pharmaceutical Use.
Benedetto Tiz D, Bagnoli L, Rosati O, Marini F, Sancineto L, Santi C.
Benedetto Tiz D, et al.
Molecules. 2022 Mar 2;27(5):1643. doi: 10.3390/molecules27051643.
Molecules. 2022.
PMID: 35268744
Free PMC article.
Review.
Item in Clipboard
Practical Synthesis and Application of Halogen-Doped Pyrrole Building Blocks.
Cotman AE, Guérin T, Kovačević I, Benedetto Tiz D, Durcik M, Fulgheri F, Možina Š, Secci D, Sterle M, Ilaš J, Zega A, Zidar N, Mašič LP, Tomašič T, Leroux FR, Hanquet G, Kikelj D.
Cotman AE, et al. Among authors: benedetto tiz d.
ACS Omega. 2021 Mar 30;6(14):9723-9730. doi: 10.1021/acsomega.1c00331. eCollection 2021 Apr 13.
ACS Omega. 2021.
PMID: 33869952
Free PMC article.
Item in Clipboard
New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity.
Durcik M, Lovison D, Skok Ž, Durante Cruz C, Tammela P, Tomašič T, Benedetto Tiz D, Draskovits G, Nyerges Á, Pál C, Ilaš J, Peterlin Mašič L, Kikelj D, Zidar N.
Durcik M, et al. Among authors: benedetto tiz d.
Eur J Med Chem. 2018 Jun 25;154:117-132. doi: 10.1016/j.ejmech.2018.05.011. Epub 2018 May 10.
Eur J Med Chem. 2018.
PMID: 29778894
Free PMC article.
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Overcoming problems of poor drug penetration into bacteria: challenges and strategies for medicinal chemists.
Benedetto Tiz D, Kikelj D, Zidar N.
Benedetto Tiz D, et al.
Expert Opin Drug Discov. 2018 Jun;13(6):497-507. doi: 10.1080/17460441.2018.1455660. Epub 2018 Mar 23.
Expert Opin Drug Discov. 2018.
PMID: 29566560
Review.
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