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Comprehensive in vitro characterization of PD-L1 small molecule inhibitors.
Sci Rep. 2019 Aug 27;9(1):12392. doi: 10.1038/s41598-019-48826-6.
Sci Rep. 2019.
PMID: 31455818
Free PMC article.
Peptidomimetic α-Acyloxymethylketone Warheads with Six-Membered Lactam P1 Glutamine Mimic: SARS-CoV-2 3CL Protease Inhibition, Coronavirus Antiviral Activity, and in Vitro Biological Stability.
Bai B, Belovodskiy A, Hena M, Kandadai AS, Joyce MA, Saffran HA, Shields JA, Khan MB, Arutyunova E, Lu J, Bajwa SK, Hockman D, Fischer C, Lamer T, Vuong W, van Belkum MJ, Gu Z, Lin F, Du Y, Xu J, Rahim M, Young HS, Vederas JC, Tyrrell DL, Lemieux MJ, Nieman JA.
Bai B, et al. Among authors: belovodskiy a.
J Med Chem. 2022 Feb 24;65(4):2905-2925. doi: 10.1021/acs.jmedchem.1c00616. Epub 2021 Jul 9.
J Med Chem. 2022.
PMID: 34242027
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Peptidomimetic nitrile warheads as SARS-CoV-2 3CL protease inhibitors.
Bai B, Arutyunova E, Khan MB, Lu J, Joyce MA, Saffran HA, Shields JA, Kandadai AS, Belovodskiy A, Hena M, Vuong W, Lamer T, Young HS, Vederas JC, Tyrrell DL, Lemieux MJ, Nieman JA.
Bai B, et al. Among authors: belovodskiy a.
RSC Med Chem. 2021 Aug 20;12(10):1722-1730. doi: 10.1039/d1md00247c. eCollection 2021 Oct 20.
RSC Med Chem. 2021.
PMID: 34778773
Free PMC article.
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Establishing normal metabolism and differentiation in hepatocellular carcinoma cells by culturing in adult human serum.
Steenbergen R, Oti M, Ter Horst R, Tat W, Neufeldt C, Belovodskiy A, Chua TT, Cho WJ, Joyce M, Dutilh BE, Tyrrell DL.
Steenbergen R, et al. Among authors: belovodskiy a.
Sci Rep. 2018 Aug 3;8(1):11685. doi: 10.1038/s41598-018-29763-2.
Sci Rep. 2018.
PMID: 30076349
Free PMC article.
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Fluorescent Hexose Conjugates Establish Stringent Stereochemical Requirement by GLUT5 for Recognition and Transport of Monosaccharides.
Soueidan OM, Scully TW, Kaur J, Panigrahi R, Belovodskiy A, Do V, Matier CD, Lemieux MJ, Wuest F, Cheeseman C, West FG.
Soueidan OM, et al. Among authors: belovodskiy a.
ACS Chem Biol. 2017 Apr 21;12(4):1087-1094. doi: 10.1021/acschembio.6b01101. Epub 2017 Mar 2.
ACS Chem Biol. 2017.
PMID: 28205432
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The Effect of Deuteration and Homologation of the Lactam Ring of Nirmatrelvir on Its Biochemical Properties and Oxidative Metabolism.
Arutyunova E, Belovodskiy A, Chen P, Khan MB, Joyce M, Saffran H, Lu J, Turner Z, Bai B, Lamer T, Young HS, Vederas JC, Tyrrell DL, Lemieux MJ, Nieman JA.
Arutyunova E, et al. Among authors: belovodskiy a.
ACS Bio Med Chem Au. 2023 Nov 15;3(6):528-541. doi: 10.1021/acsbiomedchemau.3c00039. eCollection 2023 Dec 20.
ACS Bio Med Chem Au. 2023.
PMID: 38144257
Free PMC article.
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Deuteration for Metabolic Stabilization of SARS-CoV-2 Inhibitors GC373 and Nirmatrelvir.
Van Oers TJ, Piercey A, Belovodskiy A, Reiz B, Donnelly BL, Vuong W, Lemieux MJ, Nieman JA, Auclair K, Vederas JC.
Van Oers TJ, et al. Among authors: belovodskiy a.
Org Lett. 2023 Aug 11;25(31):5885-5889. doi: 10.1021/acs.orglett.3c02140. Epub 2023 Jul 31.
Org Lett. 2023.
PMID: 37523471
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