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A Broad G Protein-Coupled Receptor Internalization Assay that Combines SNAP-Tag Labeling, Diffusion-Enhanced Resonance Energy Transfer, and a Highly Emissive Terbium Cryptate.
Front Endocrinol (Lausanne). 2015 Nov 9;6:167. doi: 10.3389/fendo.2015.00167. eCollection 2015.
Front Endocrinol (Lausanne). 2015.
PMID: 26617570
Free PMC article.
A fluorescent ligand-binding alternative using Tag-lite® technology.
Zwier JM, Roux T, Cottet M, Durroux T, Douzon S, Bdioui S, Gregor N, Bourrier E, Oueslati N, Nicolas L, Tinel N, Boisseau C, Yverneau P, Charrier-Savournin F, Fink M, Trinquet E.
Zwier JM, et al. Among authors: bdioui s.
J Biomol Screen. 2010 Dec;15(10):1248-59. doi: 10.1177/1087057110384611. Epub 2010 Oct 25.
J Biomol Screen. 2010.
PMID: 20974902
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Equilibrium Assays Are Required to Accurately Characterize the Activity Profiles of Drugs Modulating Gq-Protein-Coupled Receptors.
Bdioui S, Verdi J, Pierre N, Trinquet E, Roux T, Kenakin T.
Bdioui S, et al.
Mol Pharmacol. 2018 Sep;94(3):992-1006. doi: 10.1124/mol.118.112573. Epub 2018 Jun 28.
Mol Pharmacol. 2018.
PMID: 29954837
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The pharmacologic characterization of allosteric molecules: Gq protein activation.
Bdioui S, Verdi J, Pierre N, Trinquet E, Roux T, Kenakin T.
Bdioui S, et al.
J Recept Signal Transduct Res. 2019 Apr;39(2):106-113. doi: 10.1080/10799893.2019.1634101. Epub 2019 Jul 19.
J Recept Signal Transduct Res. 2019.
PMID: 31322035
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Nanobody-Based Quantification of GTP-Bound RHO Conformation Reveals RHOA and RHOC Activation Independent from Their Total Expression in Breast Cancer.
Keller L, Tardy C, Ligat L, Gilhodes J, Filleron T, Bery N, Rochaix P, Aquilina A, Bdioui S, Roux T, Trinquet E, Favre G, Olichon A.
Keller L, et al. Among authors: bdioui s.
Anal Chem. 2021 Apr 20;93(15):6104-6111. doi: 10.1021/acs.analchem.0c05137. Epub 2021 Apr 7.
Anal Chem. 2021.
PMID: 33825439
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