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Assessment of the Cruzain Cysteine Protease Reversible and Irreversible Covalent Inhibition Mechanism.
J Chem Inf Model. 2020 Mar 23;60(3):1666-1677. doi: 10.1021/acs.jcim.9b01138. Epub 2020 Mar 10.
J Chem Inf Model. 2020.
PMID: 32126170
Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement.
Gomes JC, Cianni L, Ribeiro J, Dos Reis Rocho F, da Costa Martins Silva S, Batista PHJ, Moraes CB, Franco CH, Freitas-Junior LHG, Kenny PW, Leitão A, Burtoloso ACB, de Vita D, Montanari CA.
Gomes JC, et al. Among authors: batista phj.
Bioorg Med Chem. 2019 Nov 15;27(22):115083. doi: 10.1016/j.bmc.2019.115083. Epub 2019 Aug 28.
Bioorg Med Chem. 2019.
PMID: 31561938
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Synthesis and matched molecular pair analysis of covalent reversible inhibitors of the cysteine protease CPB.
Matos TKB, Batista PHJ, Dos Reis Rocho F, de Vita D, Pearce N, Kellam B, Montanari CA, Leitão A.
Matos TKB, et al. Among authors: batista phj.
Bioorg Med Chem Lett. 2020 Sep 15;30(18):127439. doi: 10.1016/j.bmcl.2020.127439. Epub 2020 Jul 25.
Bioorg Med Chem Lett. 2020.
PMID: 32717373
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On the intrinsic reactivity of highly potent trypanocidal cruzain inhibitors.
Bonatto V, Batista PHJ, Cianni L, De Vita D, Silva DG, Cedron R, Tezuka DY, de Albuquerque S, Moraes CB, Franco CH, Lameira J, Leitão A, Montanari CA.
Bonatto V, et al. Among authors: batista phj.
RSC Med Chem. 2020 Sep 9;11(11):1275-1284. doi: 10.1039/d0md00097c. eCollection 2020 Nov 18.
RSC Med Chem. 2020.
PMID: 34095840
Free PMC article.
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Dipeptidyl nitrile derivatives suppress the Trypanosoma cruzi in vitro infection.
Quilles JC Jr, Shamim A, Tezuka DY, Batista PHJ, Lopes CD, de Albuquerque S, Montanari CA, Leitão A.
Quilles JC Jr, et al. Among authors: batista phj.
Exp Parasitol. 2020 Dec;219:108032. doi: 10.1016/j.exppara.2020.108032. Epub 2020 Nov 1.
Exp Parasitol. 2020.
PMID: 33137308
Free article.
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Biological Activity and Physicochemical Properties of Dipeptidyl Nitrile Derivatives Against Pancreatic Ductal Adenocarcinoma Cells.
Quilles JC Jr, Bernardi MDL, Batista PHJ, Silva SCM, Rocha CMR, Montanari CA, Leitão A.
Quilles JC Jr, et al. Among authors: batista phj.
Anticancer Agents Med Chem. 2019;19(1):112-120. doi: 10.2174/1871520618666181029141649.
Anticancer Agents Med Chem. 2019.
PMID: 30370859
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Withaferin A and Withanolide D Analogues with Dual Heat-Shock-Inducing and Cytotoxic Activities: Semisynthesis and Biological Evaluation.
Wijeratne EMK, Oliveira MCF, Mafezoli J, Xu YM, Minguzzi S, Batista PHJ, Pessoa ODL, Whitesell L, Gunatilaka AAL.
Wijeratne EMK, et al. Among authors: batista phj.
J Nat Prod. 2018 Apr 27;81(4):825-837. doi: 10.1021/acs.jnatprod.7b00918. Epub 2018 Mar 14.
J Nat Prod. 2018.
PMID: 29537263
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Withanolides from leaves of cultivated Acnistus arborescens.
Batista PH, de Lima KS, Pinto Fd, Tavares JL, de A Uchoa DE, Costa-Lotufo LV, Rocha DD, Silveira ER, Bezerra AM, Canuto KM, Pessoa OD.
Batista PH, et al.
Phytochemistry. 2016 Oct;130:321-7. doi: 10.1016/j.phytochem.2016.07.003. Epub 2016 Aug 4.
Phytochemistry. 2016.
PMID: 27498045
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