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Modifications of the Triaminoaryl Metabophore of Flupirtine and Retigabine Aimed at Avoiding Quinone Diimine Formation.
ACS Omega. 2022 Feb 25;7(9):7989-8012. doi: 10.1021/acsomega.1c07103. eCollection 2022 Mar 8.
ACS Omega. 2022.
PMID: 35284765
Free PMC article.
Carba Analogues of Flupirtine and Retigabine with Improved Oxidation Resistance and Reduced Risk of Quinoid Metabolite Formation.
Wurm KW, Bartz FM, Schulig L, Bodtke A, Bednarski PJ, Link A.
Wurm KW, et al. Among authors: bartz fm.
ChemMedChem. 2022 Aug 17;17(16):e202200262. doi: 10.1002/cmdc.202200262. Epub 2022 Jul 7.
ChemMedChem. 2022.
PMID: 35687532
Free PMC article.
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Replacing the oxidation-sensitive triaminoaryl chemotype of problematic KV 7 channel openers: Exploration of a nicotinamide scaffold.
Wurm KW, Bartz FM, Schulig L, Bodtke A, Bednarski PJ, Link A.
Wurm KW, et al. Among authors: bartz fm.
Arch Pharm (Weinheim). 2023 Feb;356(2):e2200473. doi: 10.1002/ardp.202200473. Epub 2022 Nov 17.
Arch Pharm (Weinheim). 2023.
PMID: 36395379
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A graphite furnace-atomic absorption spectrometry-based rubidium efflux assay for screening activators of the Kv 7.2/3 channel.
Bartz FM, Beirow K, Wurm K, Baecker D, Link A, Bednarski PJ.
Bartz FM, et al.
Arch Pharm (Weinheim). 2023 May;356(5):e2200585. doi: 10.1002/ardp.202200585. Epub 2023 Feb 7.
Arch Pharm (Weinheim). 2023.
PMID: 36748851
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