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Metabolism-Guided Optimization of Tryptophanol-Derived Isoindolinone p53 Activators.
Pharmaceuticals (Basel). 2023 Jan 19;16(2):146. doi: 10.3390/ph16020146.
Pharmaceuticals (Basel). 2023.
PMID: 37259297
Free PMC article.
Tryptophanol-Derived Oxazolopyrrolidone Lactams as Potential Anticancer Agents against Gastric Adenocarcinoma.
Espadinha M, Barcherini V, Gonçalves LM, Molins E, Antunes AMM, Santos MMM.
Espadinha M, et al. Among authors: barcherini v.
Pharmaceuticals (Basel). 2021 Mar 2;14(3):208. doi: 10.3390/ph14030208.
Pharmaceuticals (Basel). 2021.
PMID: 33801507
Free PMC article.
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SLMP53-2 Restores Wild-Type-Like Function to Mutant p53 through Hsp70: Promising Activity in Hepatocellular Carcinoma.
Gomes S, Bosco B, Loureiro JB, Ramos H, Raimundo L, Soares J, Nazareth N, Barcherini V, Domingues L, Oliveira C, Bisio A, Piazza S, Bauer MR, Brás JP, Almeida MI, Gomes C, Reis F, Fersht AR, Inga A, Santos MMM, Saraiva L.
Gomes S, et al. Among authors: barcherini v.
Cancers (Basel). 2019 Aug 10;11(8):1151. doi: 10.3390/cancers11081151.
Cancers (Basel). 2019.
PMID: 31405179
Free PMC article.
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SLMP53-1 interacts with wild-type and mutant p53 DNA-binding domain and reactivates multiple hotspot mutations.
Gomes AS, Ramos H, Gomes S, Loureiro JB, Soares J, Barcherini V, Monti P, Fronza G, Oliveira C, Domingues L, Bastos M, Dourado DFAR, Carvalho AL, Romão MJ, Pinheiro B, Marcelo F, Carvalho A, Santos MMM, Saraiva L.
Gomes AS, et al. Among authors: barcherini v.
Biochim Biophys Acta Gen Subj. 2020 Jan;1864(1):129440. doi: 10.1016/j.bbagen.2019.129440. Epub 2019 Sep 16.
Biochim Biophys Acta Gen Subj. 2020.
PMID: 31536751
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SLMP53-1 Inhibits Tumor Cell Growth through Regulation of Glucose Metabolism and Angiogenesis in a P53-Dependent Manner.
Ramos H, Calheiros J, Almeida J, Barcherini V, Santos S, Carvalho ATP, Santos MMM, Saraiva L.
Ramos H, et al. Among authors: barcherini v.
Int J Mol Sci. 2020 Jan 17;21(2):596. doi: 10.3390/ijms21020596.
Int J Mol Sci. 2020.
PMID: 31963392
Free PMC article.
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Potency and Selectivity Optimization of Tryptophanol-Derived Oxazoloisoindolinones: Novel p53 Activators in Human Colorectal Cancer.
Barcherini V, Almeida J, Lopes EA, Wang M, Magalhães E Silva D, Mori M, Wang S, Saraiva L, Santos MMM.
Barcherini V, et al.
ChemMedChem. 2021 Jan 8;16(1):250-258. doi: 10.1002/cmdc.202000522. Epub 2020 Sep 2.
ChemMedChem. 2021.
PMID: 32737944
Free article.
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Targeting p53 for Melanoma Treatment: Counteracting Tumour Proliferation, Dissemination and Therapeutic Resistance.
Loureiro JB, Raimundo L, Calheiros J, Carvalho C, Barcherini V, Lima NR, Gomes C, Almeida MI, Alves MG, Costa JL, Santos MMM, Saraiva L.
Loureiro JB, et al. Among authors: barcherini v.
Cancers (Basel). 2021 Apr 1;13(7):1648. doi: 10.3390/cancers13071648.
Cancers (Basel). 2021.
PMID: 33916029
Free PMC article.
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An Update on MDMX and Dual MDM2/X Inhibitors.
Espadinha M, Barcherini V, Lopes EA, Santos MMM.
Espadinha M, et al. Among authors: barcherini v.
Curr Top Med Chem. 2018;18(8):647-660. doi: 10.2174/1568026618666180604080119.
Curr Top Med Chem. 2018.
PMID: 29866007
Review.
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