Balaguer P - Search Results

1

Imidazo[2,1-b]benzothiazol Derivatives as Potential Allosteric Inhibitors of the Glucocorticoid Receptor.

Christodoulou MS, Dapiaggi F, Ghiringhelli F, Pieraccini S, Sironi M, Lucafò M, Curci D, Decorti G, Stocco G, Chirumamilla CS, Vanden Berghe W, Balaguer P, Michel BY, Burger A, Beccalli EM, Passarella D, Martinet N. Christodoulou MS, et al. Among authors: balaguer p. ACS Med Chem Lett. 2018 Feb 26;9(4):339-344. doi: 10.1021/acsmedchemlett.7b00527. eCollection 2018 Apr 12. ACS Med Chem Lett. 2018. PMID: 29670697 Free PMC article.

2

A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities.

Peiretti F, Montanari R, Capelli D, Bonardo B, Colson C, Amri EZ, Grimaldi M, Balaguer P, Ito K, Roeder RG, Pochetti G, Brunel JM. Peiretti F, et al. Among authors: balaguer p. J Med Chem. 2020 Nov 12;63(21):13124-13139. doi: 10.1021/acs.jmedchem.0c01555. Epub 2020 Nov 3. J Med Chem. 2020. PMID: 33142057 Free PMC article.

3

Structure-Based and Knowledge-Informed Design of B-Raf Inhibitors Devoid of Deleterious PXR Binding.

Schneider M, Delfosse V, Gelin M, Grimaldi M, Granell M, Heriaud L, Pons JL, Cohen Gonsaud M, Balaguer P, Bourguet W, Labesse G. Schneider M, et al. Among authors: balaguer p. J Med Chem. 2022 Jan 27;65(2):1552-1566. doi: 10.1021/acs.jmedchem.1c01354. Epub 2021 Dec 27. J Med Chem. 2022. PMID: 34958586

4

N-1H-benzimidazol-5-ylbenzenesulfonamide derivatives as potent hPXR agonists.

Benod C, Subra G, Nahoum V, Mallavialle A, Guichou JF, Milhau J, Roblés S, Bourguet W, Pascussi JM, Balaguer P, Chavanieu A. Benod C, et al. Among authors: balaguer p. Bioorg Med Chem. 2008 Apr 1;16(7):3537-49. doi: 10.1016/j.bmc.2008.02.020. Epub 2008 Feb 13. Bioorg Med Chem. 2008. PMID: 18304819

5

High Content Screening Using New U2OS Reporter Cell Models Identifies Harmol Hydrochloride as a Selective and Competitive Antagonist of the Androgen Receptor.

Dellal H, Boulahtouf A, Alaterre E, Cuenant A, Grimaldi M, Bourguet W, Gongora C, Balaguer P, Pourquier P. Dellal H, et al. Among authors: balaguer p. Cells. 2020 Jun 16;9(6):1469. doi: 10.3390/cells9061469. Cells. 2020. PMID: 32560058 Free PMC article.

6

A Comparative Study of Human and Zebrafish Pregnane X Receptor Activities of Pesticides and Steroids Using In Vitro Reporter Gene Assays.

Creusot N, Garoche C, Grimaldi M, Boulahtouf A, Chiavarina B, Bourguet W, Balaguer P. Creusot N, et al. Among authors: balaguer p. Front Endocrinol (Lausanne). 2021 May 18;12:665521. doi: 10.3389/fendo.2021.665521. eCollection 2021. Front Endocrinol (Lausanne). 2021. PMID: 34084152 Free PMC article.

7

Mutation of isoleucine 747 by a threonine alters the ligand responsiveness of the human glucocorticoid receptor.

Roux S, Térouanne B, Balaguer P, Jausons-Loffreda N, Pons M, Chambon P, Gronemeyer H, Nicolas JC. Roux S, et al. Among authors: balaguer p. Mol Endocrinol. 1996 Oct;10(10):1214-26. doi: 10.1210/mend.10.10.9121489. Mol Endocrinol. 1996. PMID: 9121489

8

Assessing the Selectivity of FXR, LXRs, CAR, and RORγ Pharmaceutical Ligands With Reporter Cell Lines.

Toporova L, Grimaldi M, Boulahtouf A, Balaguer P. Toporova L, et al. Among authors: balaguer p. Front Pharmacol. 2020 Jul 24;11:1122. doi: 10.3389/fphar.2020.01122. eCollection 2020. Front Pharmacol. 2020. PMID: 32792956 Free PMC article.

9

Molecular and Biochemical Analysis of the Estrogenic and Proliferative Properties of Vitamin E Compounds.

Khallouki F, de Medina P, Caze-Subra S, Bystricky K, Balaguer P, Poirot M, Silvente-Poirot S. Khallouki F, et al. Among authors: balaguer p. Front Oncol. 2016 Jan 5;5:287. doi: 10.3389/fonc.2015.00287. eCollection 2015. Front Oncol. 2016. PMID: 26779438 Free PMC article.

10

Assessing species-specific differences for nuclear receptor activation for environmental water extracts.

Neale PA, Grimaldi M, Boulahtouf A, Leusch FDL, Balaguer P. Neale PA, et al. Among authors: balaguer p. Water Res. 2020 Oct 15;185:116247. doi: 10.1016/j.watres.2020.116247. Epub 2020 Jul 28. Water Res. 2020. PMID: 32758789

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