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Small Molecule Kinase Inhibitor Drugs (1995-2021): Medical Indication, Pharmacology, and Synthesis.
J Med Chem. 2022 Jan 27;65(2):1047-1131. doi: 10.1021/acs.jmedchem.1c00963. Epub 2021 Oct 8.
J Med Chem. 2022.
PMID: 34624192
Free article.
Review.
Pyrazolopyrimide library screening in glioma cells discovers highly potent antiproliferative leads that target the PI3K/mTOR pathway.
Valero T, Baillache DJ, Fraser C, Myers SH, Unciti-Broceta A.
Valero T, et al. Among authors: baillache dj.
Bioorg Med Chem. 2020 Jan 1;28(1):115215. doi: 10.1016/j.bmc.2019.115215. Epub 2019 Nov 25.
Bioorg Med Chem. 2020.
PMID: 31787462
Free PMC article.
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Recent developments in anticancer kinase inhibitors based on the pyrazolo[3,4-d]pyrimidine scaffold.
Baillache DJ, Unciti-Broceta A.
Baillache DJ, et al.
RSC Med Chem. 2020 Sep 8;11(10):1112-1135. doi: 10.1039/d0md00227e. eCollection 2020 Oct 1.
RSC Med Chem. 2020.
PMID: 33479617
Free PMC article.
Review.
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A 5-FU Precursor Designed to Evade Anabolic and Catabolic Drug Pathways and Activated by Pd Chemistry In Vitro and In Vivo.
Adam C, Bray TL, Pérez-López AM, Tan EH, Rubio-Ruiz B, Baillache DJ, Houston DR, Salji MJ, Leung HY, Unciti-Broceta A.
Adam C, et al. Among authors: baillache dj.
J Med Chem. 2022 Jan 13;65(1):552-561. doi: 10.1021/acs.jmedchem.1c01733. Epub 2022 Jan 3.
J Med Chem. 2022.
PMID: 34979089
Free article.
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The Design of Potent, Selective and Drug-Like RGD αvβ1 Small-Molecule Inhibitors Derived from non-RGD α4β1 Antagonists.
Hatley RJD, Barrett TN, Slack RJ, Watson ME, Baillache DJ, Gruszka A, Washio Y, Rowedder JE, Pogány P, Pal S, Macdonald SJF.
Hatley RJD, et al. Among authors: baillache dj.
ChemMedChem. 2019 Jul 17;14(14):1315-1320. doi: 10.1002/cmdc.201900359. Epub 2019 Jul 1.
ChemMedChem. 2019.
PMID: 31207080
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Discovery of pyrazolopyrimidines that selectively inhibit CSF-1R kinase by iterative design, synthesis and screening against glioblastoma cells.
Baillache DJ, Valero T, Lorente-Macías Á, Bennett DJ, Elliott RJR, Carragher NO, Unciti-Broceta A.
Baillache DJ, et al.
RSC Med Chem. 2023 Oct 11;14(12):2611-2624. doi: 10.1039/d3md00454f. eCollection 2023 Dec 13.
RSC Med Chem. 2023.
PMID: 38099057
Free PMC article.
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