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Synthesis and structure-activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis.
J Enzyme Inhib Med Chem. 2018 Dec;33(1):1271-1282. doi: 10.1080/14756366.2018.1490731.
J Enzyme Inhib Med Chem. 2018.
PMID: 30230387
Free PMC article.
Synthesis and in vitro pharmacological evaluation of N-[(1-benzyl-1,2,3-triazol-4-yl)methyl]-carboxamides on d-secoestrone scaffolds.
Szabó J, Bacsa I, Wölfling J, Schneider G, Zupkó I, Varga M, Herman BE, Kalmár L, Szécsi M, Mernyák E.
Szabó J, et al. Among authors: bacsa i.
J Enzyme Inhib Med Chem. 2016 Aug;31(4):574-9. doi: 10.3109/14756366.2015.1050008. Epub 2015 Sep 11.
J Enzyme Inhib Med Chem. 2016.
PMID: 26360618
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Synthesis of A-ring halogenated 13α-estrone derivatives as potential 17β-HSD1 inhibitors.
Bacsa I, Jójárt R, Schneider G, Wölfling J, Maróti P, Herman BE, Szécsi M, Mernyák E.
Bacsa I, et al.
Steroids. 2015 Dec;104:230-6. doi: 10.1016/j.steroids.2015.10.008. Epub 2015 Oct 22.
Steroids. 2015.
PMID: 26476182
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Comparative investigation of the in vitro inhibitory potencies of 13-epimeric estrones and D-secoestrones towards 17β-hydroxysteroid dehydrogenase type 1.
Herman BE, Szabó J, Bacsa I, Wölfling J, Schneider G, Bálint M, Hetényi C, Mernyák E, Szécsi M.
Herman BE, et al. Among authors: bacsa i.
J Enzyme Inhib Med Chem. 2016;31(sup3):61-69. doi: 10.1080/14756366.2016.1204610. Epub 2016 Jul 18.
J Enzyme Inhib Med Chem. 2016.
PMID: 27424610
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Synthesis of novel 13α-estrone derivatives by Sonogashira coupling as potential 17β-HSD1 inhibitors.
Bacsa I, Jójárt R, Wölfling J, Schneider G, Herman BE, Szécsi M, Mernyák E.
Bacsa I, et al.
Beilstein J Org Chem. 2017 Jun 30;13:1303-1309. doi: 10.3762/bjoc.13.126. eCollection 2017.
Beilstein J Org Chem. 2017.
PMID: 28694873
Free PMC article.
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The first Pd-catalyzed Buchwald-Hartwig aminations at C-2 or C-4 in the estrone series.
Bacsa I, Szemerédi D, Wölfling J, Schneider G, Fekete L, Mernyák E.
Bacsa I, et al.
Beilstein J Org Chem. 2018 May 4;14:998-1003. doi: 10.3762/bjoc.14.85. eCollection 2018.
Beilstein J Org Chem. 2018.
PMID: 29977371
Free PMC article.
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Syntheses and antiproliferative effects of D-homo- and D-secoestrones.
Mernyák E, Szabó J, Bacsa I, Huber J, Schneider G, Minorics R, Bózsity N, Zupkó I, Varga M, Bikádi Z, Hazai E, Wölfling J.
Mernyák E, et al. Among authors: bacsa i.
Steroids. 2014 Sep;87:128-36. doi: 10.1016/j.steroids.2014.05.015. Epub 2014 Jun 10.
Steroids. 2014.
PMID: 24928727
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Synthesis of Novel C-2- or C-15-Labeled BODIPY-Estrone Conjugates.
Bacsa I, Konc C, Orosz AB, Kecskeméti G, Rigó R, Özvegy-Laczka C, Mernyák E.
Bacsa I, et al.
Molecules. 2018 Apr 3;23(4):821. doi: 10.3390/molecules23040821.
Molecules. 2018.
PMID: 29614041
Free PMC article.
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