Highly efficient asymmetric synthesis of sitagliptin.
Hansen KB, Hsiao Y, Xu F, Rivera N, Clausen A, Kubryk M, Krska S, Rosner T, Simmons B, Balsells J, Ikemoto N, Sun Y, Spindler F, Malan C, Grabowski EJ, Armstrong JD 3rd.
Hansen KB, et al. Among authors: armstrong jd 3rd.
J Am Chem Soc. 2009 Jul 1;131(25):8798-804. doi: 10.1021/ja902462q.
J Am Chem Soc. 2009.
PMID: 19507853