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Lead Optimization of Benzoxazolone Carboxamides as Orally Bioavailable and CNS Penetrant Acid Ceramidase Inhibitors.
Di Martino S, Tardia P, Cilibrasi V, Caputo S, Mazzonna M, Russo D, Penna I, Realini N, Margaroli N, Migliore M, Pizzirani D, Ottonello G, Bertozzi SM, Armirotti A, Nguyen D, Sun Y, Bongarzone ER, Lansbury P, Liu M, Skerlj R, Scarpelli R. Di Martino S, et al. Among authors: armirotti a. J Med Chem. 2020 Apr 9;63(7):3634-3664. doi: 10.1021/acs.jmedchem.9b02004. Epub 2020 Mar 26. J Med Chem. 2020. PMID: 32176488 Free PMC article.
beta-amyloid is different in normal aging and in Alzheimer disease.
Piccini A, Russo C, Gliozzi A, Relini A, Vitali A, Borghi R, Giliberto L, Armirotti A, D'Arrigo C, Bachi A, Cattaneo A, Canale C, Torrassa S, Saido TC, Markesbery W, Gambetti P, Tabaton M. Piccini A, et al. Among authors: armirotti a. J Biol Chem. 2005 Oct 7;280(40):34186-92. doi: 10.1074/jbc.M501694200. Epub 2005 Aug 15. J Biol Chem. 2005. PMID: 16103127 Free article.
5-fluorouracil causes endothelial cell senescence: potential protective role of glucagon-like peptide 1.
Altieri P, Murialdo R, Barisione C, Lazzarini E, Garibaldi S, Fabbi P, Ruggeri C, Borile S, Carbone F, Armirotti A, Canepa M, Ballestrero A, Brunelli C, Montecucco F, Ameri P, Spallarossa P. Altieri P, et al. Among authors: armirotti a. Br J Pharmacol. 2017 Nov;174(21):3713-3726. doi: 10.1111/bph.13725. Epub 2017 Feb 22. Br J Pharmacol. 2017. PMID: 28127745 Free PMC article.
Downregulation of myosin II-B by siRNA alters the subcellular localization of the amyloid precursor protein and increases amyloid-beta deposition in N2a cells.
Massone S, Argellati F, Passalacqua M, Armirotti A, Melone L, d'Abramo C, Marinari UM, Domenicotti C, Pronzato MA, Ricciarelli R. Massone S, et al. Among authors: armirotti a. Biochem Biophys Res Commun. 2007 Oct 26;362(3):633-8. doi: 10.1016/j.bbrc.2007.08.061. Epub 2007 Aug 21. Biochem Biophys Res Commun. 2007. PMID: 17727819
ADP-ribosyl cyclases generate two unusual adenine homodinucleotides with cytotoxic activity on mammalian cells.
Basile G, Taglialatela-Scafati O, Damonte G, Armirotti A, Bruzzone S, Guida L, Franco L, Usai C, Fattorusso E, De Flora A, Zocchi E. Basile G, et al. Among authors: armirotti a. Proc Natl Acad Sci U S A. 2005 Oct 11;102(41):14509-14. doi: 10.1073/pnas.0503691102. Epub 2005 Sep 19. Proc Natl Acad Sci U S A. 2005. PMID: 16172408 Free PMC article.
139 results