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An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library.
Eur J Med Chem. 2024 Apr 15;270:116362. doi: 10.1016/j.ejmech.2024.116362. Epub 2024 Mar 28.
Eur J Med Chem. 2024.
PMID: 38574637
The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas.
Ardino C, Sannio F, Pasero C, Botta L, Dreassi E, Docquier JD, D'Agostino I.
Ardino C, et al.
Mol Divers. 2023 Jun;27(3):1489-1499. doi: 10.1007/s11030-022-10505-6. Epub 2022 Aug 29.
Mol Divers. 2023.
PMID: 36036302
Free PMC article.
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Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA.
D'Agostino I, Ardino C, Poli G, Sannio F, Lucidi M, Poggialini F, Visaggio D, Rango E, Filippi S, Petricci E, Visca P, Botta L, Docquier JD, Dreassi E.
D'Agostino I, et al. Among authors: ardino c.
Eur J Med Chem. 2022 Mar 5;231:114158. doi: 10.1016/j.ejmech.2022.114158. Epub 2022 Jan 29.
Eur J Med Chem. 2022.
PMID: 35168113
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