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Discovery and SAR of JTE-151: A Novel RORγ Inhibitor for Clinical Development.
J Med Chem. 2024 Jan 25;67(2):952-970. doi: 10.1021/acs.jmedchem.3c01933. Epub 2024 Jan 3.
J Med Chem. 2024.
PMID: 38170624
Indirubin, a component of Ban-Lan-Gen, activates CYP3A4 gene transcription through the human pregnane X receptor.
Kumagai T, Aratsu Y, Sugawara R, Sasaki T, Miyairi S, Nagata K.
Kumagai T, et al. Among authors: aratsu y.
Drug Metab Pharmacokinet. 2016 Apr;31(2):139-45. doi: 10.1016/j.dmpk.2016.01.002. Epub 2016 Jan 22.
Drug Metab Pharmacokinet. 2016.
PMID: 26987505
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SAR Exploration Guided by LE and Fsp(3): Discovery of a Selective and Orally Efficacious RORγ Inhibitor.
Hirata K, Kotoku M, Seki N, Maeba T, Maeda K, Hirashima S, Sakai T, Obika S, Hori A, Hase Y, Yamaguchi T, Katsuda Y, Hata T, Miyagawa N, Arita K, Nomura Y, Asahina K, Aratsu Y, Kamada M, Adachi T, Noguchi M, Doi S, Crowe P, Bradley E, Steensma R, Tao H, Fenn M, Babine R, Li X, Thacher S, Hashimoto H, Shiozaki M.
Hirata K, et al. Among authors: aratsu y.
ACS Med Chem Lett. 2015 Nov 4;7(1):23-7. doi: 10.1021/acsmedchemlett.5b00253. eCollection 2016 Jan 14.
ACS Med Chem Lett. 2015.
PMID: 26819660
Free PMC article.
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JTP-103237, a novel monoacylglycerol acyltransferase inhibitor, modulates fat absorption and prevents diet-induced obesity.
Okuma C, Ohta T, Tadaki H, Hamada H, Oda T, Taniuchi H, Yamanaka K, Ishii Y, Ohe Y, Yata S, Nishiu J, Aratsu Y, Oshida S, Kume S, Kakutani M.
Okuma C, et al. Among authors: aratsu y.
Eur J Pharmacol. 2015 Jul 5;758:72-81. doi: 10.1016/j.ejphar.2015.03.072. Epub 2015 Apr 6.
Eur J Pharmacol. 2015.
PMID: 25857225
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Unveiling a new essential cis element for the transactivation of the CYP3A4 gene by xenobiotics.
Toriyabe T, Nagata K, Takada T, Aratsu Y, Matsubara T, Yoshinari K, Yamazoe Y.
Toriyabe T, et al. Among authors: aratsu y.
Mol Pharmacol. 2009 Mar;75(3):677-84. doi: 10.1124/mol.108.050575. Epub 2008 Dec 15.
Mol Pharmacol. 2009.
PMID: 19074998
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