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BCAAs and Di-Alanine supplementation in the prevention of skeletal muscle atrophy: preclinical evaluation in a murine model of hind limb unloading.
Mantuano P, Boccanegra B, Bianchini G, Conte E, De Bellis M, Sanarica F, Camerino GM, Pierno S, Cappellari O, Allegretti M, Aramini A, De Luca A. Mantuano P, et al. Among authors: aramini a. Pharmacol Res. 2021 Sep;171:105798. doi: 10.1016/j.phrs.2021.105798. Epub 2021 Aug 2. Pharmacol Res. 2021. PMID: 34352400
Design of noncompetitive interleukin-8 inhibitors acting on CXCR1 and CXCR2.
Moriconi A, Cesta MC, Cervellera MN, Aramini A, Coniglio S, Colagioia S, Beccari AR, Bizzarri C, Cavicchia MR, Locati M, Galliera E, Di Benedetto P, Vigilante P, Bertini R, Allegretti M. Moriconi A, et al. Among authors: aramini a. J Med Chem. 2007 Aug 23;50(17):3984-4002. doi: 10.1021/jm061469t. Epub 2007 Aug 1. J Med Chem. 2007. PMID: 17665889
Development and validation of an LC-MS/MS method for determination of methanesulfonamide in human urine.
Anacardio R, Mullins FG, Hannam S, Sheikh MS, O'Shea K, Aramini A, D'Anniballe G, D'Anteo L, Ferrari MP, Allegretti M. Anacardio R, et al. Among authors: aramini a. J Chromatogr B Analyt Technol Biomed Life Sci. 2009 Jul 15;877(22):2087-92. doi: 10.1016/j.jchromb.2009.05.051. Epub 2009 Jun 17. J Chromatogr B Analyt Technol Biomed Life Sci. 2009. PMID: 19539545
Structure-Activity Relationship of novel phenylacetic CXCR1 inhibitors.
Sablone MR, Cesta MC, Moriconi A, Aramini A, Bizzarri C, Di Giacinto C, Di Bitondo R, Gloaguen I, Aschi M, Crucianelli M, Bertini R, Allegretti M. Sablone MR, et al. Among authors: aramini a. Bioorg Med Chem Lett. 2009 Aug 1;19(15):4026-30. doi: 10.1016/j.bmcl.2009.06.027. Epub 2009 Jun 13. Bioorg Med Chem Lett. 2009. PMID: 19560921
Receptor binding mode and pharmacological characterization of a potent and selective dual CXCR1/CXCR2 non-competitive allosteric inhibitor.
Bertini R, Barcelos LS, Beccari AR, Cavalieri B, Moriconi A, Bizzarri C, Di Benedetto P, Di Giacinto C, Gloaguen I, Galliera E, Corsi MM, Russo RC, Andrade SP, Cesta MC, Nano G, Aramini A, Cutrin JC, Locati M, Allegretti M, Teixeira MM. Bertini R, et al. Among authors: aramini a. Br J Pharmacol. 2012 Jan;165(2):436-54. doi: 10.1111/j.1476-5381.2011.01566.x. Br J Pharmacol. 2012. PMID: 21718305 Free PMC article.
Targeting the minor pocket of C5aR for the rational design of an oral allosteric inhibitor for inflammatory and neuropathic pain relief.
Moriconi A, Cunha TM, Souza GR, Lopes AH, Cunha FQ, Carneiro VL, Pinto LG, Brandolini L, Aramini A, Bizzarri C, Bianchini G, Beccari AR, Fanton M, Bruno A, Costantino G, Bertini R, Galliera E, Locati M, Ferreira SH, Teixeira MM, Allegretti M. Moriconi A, et al. Among authors: aramini a. Proc Natl Acad Sci U S A. 2014 Nov 25;111(47):16937-42. doi: 10.1073/pnas.1417365111. Epub 2014 Nov 10. Proc Natl Acad Sci U S A. 2014. PMID: 25385614 Free PMC article.
DFL23448, A Novel Transient Receptor Potential Melastin 8-Selective Ion Channel Antagonist, Modifies Bladder Function and Reduces Bladder Overactivity in Awake Rats.
Mistretta FA, Russo A, Castiglione F, Bettiga A, Colciago G, Montorsi F, Brandolini L, Aramini A, Bianchini G, Allegretti M, Bovolenta S, Russo R, Benigni F, Hedlund P. Mistretta FA, et al. Among authors: aramini a. J Pharmacol Exp Ther. 2016 Jan;356(1):200-11. doi: 10.1124/jpet.115.228684. Epub 2015 Nov 6. J Pharmacol Exp Ther. 2016. PMID: 26546575
44 results