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Imidazopyridine-fused [1,3]-diazepinones: synthesis and antiproliferative activity.
Eur J Med Chem. 2014 Mar 21;75:382-90. doi: 10.1016/j.ejmech.2014.01.044. Epub 2014 Jan 30.
Eur J Med Chem. 2014.
PMID: 24561668
Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7.
Arama DP, Soualmia F, Lisowski V, Longevial JF, Bosc E, Maillard LT, Martinez J, Masurier N, El Amri C.
Arama DP, et al.
Eur J Med Chem. 2015 Mar 26;93:202-13. doi: 10.1016/j.ejmech.2015.02.008. Epub 2015 Feb 7.
Eur J Med Chem. 2015.
PMID: 25682203
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Imidazopyridine-fused [1,3]-diazepinones part 2: Structure-activity relationships and antiproliferative activity against melanoma cells.
Bellet V, Lichon L, Arama DP, Gallud A, Lisowski V, Maillard LT, Garcia M, Martinez J, Masurier N.
Bellet V, et al. Among authors: arama dp.
Eur J Med Chem. 2017 Jan 5;125:1225-1234. doi: 10.1016/j.ejmech.2016.11.023. Epub 2016 Nov 11.
Eur J Med Chem. 2017.
PMID: 27871038
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Inhibitors of kallikrein-related peptidases: An overview.
Masurier N, Arama DP, El Amri C, Lisowski V.
Masurier N, et al. Among authors: arama dp.
Med Res Rev. 2018 Mar;38(2):655-683. doi: 10.1002/med.21451. Epub 2017 Jun 13.
Med Res Rev. 2018.
PMID: 28609548
Review.
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Identification of Quinazolinone Analogs Targeting CDK5 Kinase Activity and Glioblastoma Cell Proliferation.
Peyressatre M, Arama DP, Laure A, González-Vera JA, Pellerano M, Masurier N, Lisowski V, Morris MC.
Peyressatre M, et al. Among authors: arama dp.
Front Chem. 2020 Aug 19;8:691. doi: 10.3389/fchem.2020.00691. eCollection 2020.
Front Chem. 2020.
PMID: 32974274
Free PMC article.
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