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Page 1
Meldrum's acid derivates are MepA efflux pump inhibitors: In vitro and in silico essays.
Araújo IM, Pereira RLS, de Araújo ACJ, Gonçalves SA, Tintino SR, Oliveira-Tintino CDM, de Menezes IRA, Salamoni R, Begnini IM, Rebelo RA, Silva LED, Gurgel APAD, Coutinho HDM. Araújo IM, et al. Among authors: de araujo acj. J Basic Microbiol. 2024 Feb;64(2):e2300558. doi: 10.1002/jobm.202300558. Epub 2023 Dec 18. J Basic Microbiol. 2024. PMID: 38110852
Chemical composition and antibacterial effects of Etlingera elatior (Jack) R.M. Smith against Staphylococcus aureus efflux pumps.
de Sousa Ferreira F, de Araújo Neto JB, de Morais Oliveira-Tintino CD, de Araújo ACJ, Ribeiro-Filho J, Freitas PR, Araújo IM, Lima MA, de Azevedo FR, Tintino SR, Coutinho HDM, Navarro DMDAF. de Sousa Ferreira F, et al. Among authors: de araujo acj. Chem Biol Interact. 2023 Dec 1;386:110751. doi: 10.1016/j.cbi.2023.110751. Epub 2023 Oct 10. Chem Biol Interact. 2023. PMID: 37821044
Potentiating-antibiotic activity and absorption, distribution, metabolism, excretion and toxicity properties (ADMET) analysis of synthetic thiadiazines against multi-drug resistant (MDR) strains.
de Araújo ACJ, Freitas PR, Araújo IM, Siqueira GM, de Oliveira Borges JA, Alves DS, Miranda GM, Dos Santos Nascimento IJ, de Araújo-Júnior JX, da Silva-Júnior EF, de Aquino TM, Junior FJBM, Marinho ES, Dos Santos HS, Tintino SR, Coutinho HDM. de Araújo ACJ, et al. Fundam Clin Pharmacol. 2024 Feb;38(1):84-98. doi: 10.1111/fcp.12950. Epub 2023 Aug 30. Fundam Clin Pharmacol. 2024. PMID: 37649138
Synthesis, spectroscopic characterization, and antibacterial activity of chalcone (2E)-1-(3'-aminophenyl)-3-(4-dimethylaminophenyl)-prop-2-en-1-one against multiresistant Staphylococcus aureus carrier of efflux pump mechanisms and β-lactamase.
da Silva L, Donato IA, Bezerra SR, Dos Santos HS, Bandeira PN, do Nascimento MTR, Guedes JM, Freitas PR, de Araújo ACJ, de Freitas TS, Coutinho HDM, de Matos YMLS, de Oliveira LCC, da Cunha FAB. da Silva L, et al. Among authors: de araujo acj. Fundam Clin Pharmacol. 2024 Feb;38(1):60-71. doi: 10.1111/fcp.12938. Epub 2023 Jul 27. Fundam Clin Pharmacol. 2024. PMID: 37497790
Antibiotic-Potentiating Activity of the Schinus terebinthifolius Raddi Essential Oil against MDR Bacterial Strains.
Costa da Silva MM, Bezerra de Araújo Neto J, Lucas Dos Santos AT, de Morais Oliveira-Tintino CD, de Araújo ACJ, Freitas PR, da Silva LE, do Amaral W, Deschamps C, de Azevedo FR, Gonçalves Lima CM, Golubkina N, Calixto-Júnior JT, Ribeiro-Filho J, Coutinho HDM, Caruso G, Tintino SR. Costa da Silva MM, et al. Among authors: de araujo acj. Plants (Basel). 2023 Apr 8;12(8):1587. doi: 10.3390/plants12081587. Plants (Basel). 2023. PMID: 37111810 Free PMC article.
Terpenes as bacterial efflux pump inhibitors: A systematic review.
Dias KJSO, Miranda GM, Bessa JR, Araújo ACJ, Freitas PR, Almeida RS, Paulo CLR, Neto JBA, Coutinho HDM, Ribeiro-Filho J. Dias KJSO, et al. Among authors: araujo acj. Front Pharmacol. 2022 Oct 13;13:953982. doi: 10.3389/fphar.2022.953982. eCollection 2022. Front Pharmacol. 2022. PMID: 36313340 Free PMC article.
Ferulic acid derivatives inhibiting Staphylococcus aureus tetK and MsrA efflux pumps.
Pinheiro PG, Santiago GMP, da Silva FEF, de Araújo ACJ, de Oliveira CRT, Freitas PR, Rocha JE, Neto JBA, da Silva MMC, Tintino SR, Siyadatpanah A, Norouzi R, Dashti S, Wilairatana P, Coutinho HDM, da Costa JGM. Pinheiro PG, et al. Among authors: de araujo acj. Biotechnol Rep (Amst). 2022 Mar 4;34:e00717. doi: 10.1016/j.btre.2022.e00717. eCollection 2022 Jun. Biotechnol Rep (Amst). 2022. PMID: 35284249 Free PMC article.
Enhancement of the antibiotic activity mediated by the essential oil of Ocotea odorifera (VELL) ROWHER and safrole association.
de Almeida RS, Ribeiro-Filho J, Freitas PR, de Araújo ACJ, Dos Santos EL, Tintino SR, Moura TF, Ferreira VA, Ferreira BA, Juno Alencar Fonseca V, Leite PIP, Albuquerque da Silva AC, Everson da Silva L, do Amaral W, Deschamps C, Siyadatpanah A, Wilairatana P, Coutinho HDM. de Almeida RS, et al. Among authors: de araujo acj. J Infect Public Health. 2022 Mar;15(3):373-377. doi: 10.1016/j.jiph.2021.09.028. Epub 2021 Oct 7. J Infect Public Health. 2022. PMID: 34656506 Free article.
Characterization and Evaluation of Layered Bi2WO6 Nanosheets as a New Antibacterial Agent.
Leandro MKDNS, Moura JVB, Freire PTC, Vega ML, Lima CDL, Hidalgo ÁA, Araújo ACJ, Freitas PR, Paulo CLR, Sousa AK, Rocha JE, Leandro LMG, Silva ROMD, Cruz-Martins N, Coutinho HDM. Leandro MKDNS, et al. Among authors: araujo acj. Antibiotics (Basel). 2021 Sep 3;10(9):1068. doi: 10.3390/antibiotics10091068. Antibiotics (Basel). 2021. PMID: 34572651 Free PMC article.
Inhibition of the MepA efflux pump by limonene demonstrated by in vitro and in silico methods.
Freitas PR, de Araújo ACJ, Dos Santos Barbosa CR, Muniz DF, de Almeida RS, de Menezes IRA, da Costa JGM, Rodrigues FFG, Rocha JE, Pereira-Junior FN, Tintino SR, Coutinho HDM. Freitas PR, et al. Among authors: de araujo acj. Folia Microbiol (Praha). 2022 Feb;67(1):15-20. doi: 10.1007/s12223-021-00909-6. Epub 2021 Aug 20. Folia Microbiol (Praha). 2022. PMID: 34417720
21 results