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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
---|---|
2014 | 1 |
2016 | 4 |
2017 | 1 |
2024 | 0 |
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6 results
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Page 1
A Fluorescent-Labeled Phosphono Bisbenzguanidine As an Activity-Based Probe for Matriptase.
Chemistry. 2017 Apr 19;23(22):5205-5209. doi: 10.1002/chem.201700319. Epub 2017 Mar 28.
Chemistry. 2017.
PMID: 28370501
Evaluation of bisbenzamidines as inhibitors for matriptase-2.
Beckmann AM, Gilberg E, Gattner S, Huang TL, Vanden Eynde JJ, Mayence A, Bajorath J, Stirnberg M, Gütschow M.
Beckmann AM, et al.
Bioorg Med Chem Lett. 2016 Aug 1;26(15):3741-5. doi: 10.1016/j.bmcl.2016.05.071. Epub 2016 May 26.
Bioorg Med Chem Lett. 2016.
PMID: 27287367
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The intact Kunitz domain protects the amyloid precursor protein from being processed by matriptase-2.
Beckmann AM, Glebov K, Walter J, Merkel O, Mangold M, Schmidt F, Becker-Pauly C, Gütschow M, Stirnberg M.
Beckmann AM, et al.
Biol Chem. 2016 Aug 1;397(8):777-90. doi: 10.1515/hsz-2015-0263.
Biol Chem. 2016.
PMID: 27078672
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3,1-Benzothiazines, 1,4-Benzodioxines and 1,4-Benzoxazines as Inhibitors of Matriptase-2: Outcome of a Focused Screening Approach.
Roydeva PG, Beckmann AM, Stirnberg M, Cesar J, Kikelj D, Ilaš J, Gütschow M.
Roydeva PG, et al. Among authors: beckmann am.
Pharmaceuticals (Basel). 2016 Jan 13;9(1):2. doi: 10.3390/ph9010002.
Pharmaceuticals (Basel). 2016.
PMID: 26771619
Free PMC article.
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En Route to New Therapeutic Options for Iron Overload Diseases: Matriptase-2 as a Target for Kunitz-Type Inhibitors.
Beckmann AM, Maurer E, Lülsdorff V, Wilms A, Furtmann N, Bajorath J, Gütschow M, Stirnberg M.
Beckmann AM, et al.
Chembiochem. 2016 Apr 1;17(7):595-604. doi: 10.1002/cbic.201500651. Epub 2016 Feb 16.
Chembiochem. 2016.
PMID: 26762582
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3-Cyano-3-aza-β-amino Acid Derivatives as Inhibitors of Human Cysteine Cathepsins.
Schmitz J, Beckmann AM, Dudic A, Li T, Sellier R, Bartz U, Gütschow M.
Schmitz J, et al. Among authors: beckmann am.
ACS Med Chem Lett. 2014 Aug 11;5(10):1076-81. doi: 10.1021/ml500238q. eCollection 2014 Oct 9.
ACS Med Chem Lett. 2014.
PMID: 25313316
Free PMC article.
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