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Year Number of Results
2015 2
2016 5
2017 15
2018 25
2019 46
2020 48
2021 39
2022 40
2023 30
2024 6

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229 results

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Page 1
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction.
Giovannuzzi S, Chavarria D, Provensi G, Leri M, Bucciantini M, Carradori S, Bonardi A, Gratteri P, Borges F, Nocentini A, Supuran CT. Giovannuzzi S, et al. Among authors: nocentini a. J Med Chem. 2024 Mar 14;67(5):4170-4193. doi: 10.1021/acs.jmedchem.4c00045. Epub 2024 Mar 4. J Med Chem. 2024. PMID: 38436571
Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases.
Fuentes-Aguilar A, González-Bakker A, Jovanović M, Stojanov SJ, Puerta A, Gargano A, Dinić J, Vega-Báez JL, Merino-Montiel P, Montiel-Smith S, Alcaro S, Nocentini A, Pešić M, Supuran CT, Padrón JM, Fernández-Bolaños JG, López Ó. Fuentes-Aguilar A, et al. Among authors: nocentini a. Bioorg Chem. 2024 Apr;145:107168. doi: 10.1016/j.bioorg.2024.107168. Epub 2024 Feb 6. Bioorg Chem. 2024. PMID: 38354500 Free article.
Boron-containing carbonic anhydrases inhibitors.
Giovannuzzi S, Nikitjuka A, Pereira Resende BR, Smietana M, Nocentini A, Supuran CT, Winum JY. Giovannuzzi S, et al. Among authors: nocentini a. Bioorg Chem. 2024 Feb;143:106976. doi: 10.1016/j.bioorg.2023.106976. Epub 2023 Nov 19. Bioorg Chem. 2024. PMID: 38000350 Review.
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates.
Giovannuzzi S, Marapaka AK, Abutaleb NS, Carta F, Liang HW, Nocentini A, Pisano L, Seleem MN, Flaherty DP, Supuran CT. Giovannuzzi S, et al. Among authors: nocentini a. J Enzyme Inhib Med Chem. 2023 Dec;38(1):2284119. doi: 10.1080/14756366.2023.2284119. Epub 2023 Nov 23. J Enzyme Inhib Med Chem. 2023. PMID: 37994421 Free PMC article.
4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activity against Multidrug Resistant Cancer Cells.
Masci D, Puxeddu M, Di Magno L, D'Ambrosio M, Parisi A, Nalli M, Bai R, Coluccia A, Sciò P, Orlando V, D'Angelo S, Biagioni S, Urbani A, Hamel E, Nocentini A, Filiberti S, Turati M, Ronca R, Kopecka J, Riganti C, Fionda C, Bordone R, Della Rocca G, Canettieri G, Supuran CT, Silvestri R, La Regina G. Masci D, et al. Among authors: nocentini a. J Med Chem. 2023 Nov 9;66(21):14824-14842. doi: 10.1021/acs.jmedchem.3c01424. Epub 2023 Oct 30. J Med Chem. 2023. PMID: 37902628 Free PMC article.
Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold.
Romagnoli R, De Ventura T, Manfredini S, Baldini E, Supuran CT, Nocentini A, Brancale A, Bortolozzi R, Manfreda L, Viola G. Romagnoli R, et al. Among authors: nocentini a. J Enzyme Inhib Med Chem. 2023 Dec;38(1):2270180. doi: 10.1080/14756366.2023.2270180. Epub 2023 Oct 18. J Enzyme Inhib Med Chem. 2023. PMID: 37850364 Free PMC article.
229 results