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Page 1
Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates.
Machulkin AE, Skvortsov DA, Ivanenkov YA, Ber AP, Kavalchuk MV, Aladinskaya AV, Uspenskaya AA, Shafikov RR, Plotnikova EA, Yakubovskaya RI, Nimenko EA, Zyk NU, Beloglazkina EK, Zyk NV, Koteliansky VE, Majouga AG. Machulkin AE, et al. Among authors: aladinskaya av. Bioorg Med Chem Lett. 2019 Aug 15;29(16):2229-2235. doi: 10.1016/j.bmcl.2019.06.035. Epub 2019 Jun 20. Bioorg Med Chem Lett. 2019. PMID: 31248772
Small-molecule PSMA ligands. Current state, SAR and perspectives.
Machulkin AE, Ivanenkov YA, Aladinskaya AV, Veselov MS, Aladinskiy VA, Beloglazkina EK, Koteliansky VE, Shakhbazyan AG, Sandulenko YB, Majouga AG. Machulkin AE, et al. Among authors: aladinskaya av. J Drug Target. 2016 Sep;24(8):679-93. doi: 10.3109/1061186X.2016.1154564. Epub 2016 Mar 10. J Drug Target. 2016. PMID: 26887438 Review.
Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA.
Ivanenkov YA, Machulkin AE, Garanina AS, Skvortsov DA, Uspenskaya AA, Deyneka EV, Trofimenko AV, Beloglazkina EK, Zyk NV, Koteliansky VE, Bezrukov DS, Aladinskaya AV, Vorobyeva NS, Puchinina MM, Riabykh GK, Sofronova AA, Malyshev AS, Majouga AG. Ivanenkov YA, et al. Among authors: aladinskaya av. Bioorg Med Chem Lett. 2019 May 15;29(10):1246-1255. doi: 10.1016/j.bmcl.2019.01.040. Epub 2019 Feb 1. Bioorg Med Chem Lett. 2019. PMID: 30904185
Corrigendum to 'Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA' [Bioor. Med. Chem. Lett. 29/10 (2019) 1246-1255].
Ivanenkov YA, Machulkin AE, Garanina AS, Skvortsov DA, Uspenskaya AA, Deyneka EV, Trofimenko AV, Beloglazkina EK, Zyk NV, Koteliansky VE, Bezrukov DS, Aladinskaya AV, Vorobyeva NS, Puchinina MM, Ryabykh GK, Sofronova AA, Malyshev AS, Majouga AG. Ivanenkov YA, et al. Among authors: aladinskaya av. Bioorg Med Chem Lett. 2019 Jul 1;29(13):1688. doi: 10.1016/j.bmcl.2019.04.038. Epub 2019 May 2. Bioorg Med Chem Lett. 2019. PMID: 31056242 No abstract available.
In Silico Approaches to the Design of NS5A Inhibitors.
Ivanenkov YA, Veselov MS, Aladinskiy VA, Shakhbazyan AG, Yartseva SM, Majouga AG, Aladinskaya AV, Vantskul AS, Leonov SV, Ivachtchenko AV, Koteliansky VE. Ivanenkov YA, et al. Among authors: aladinskaya av. Curr Top Med Chem. 2016;16(12):1383-91. doi: 10.2174/1568026616666151120113705. Curr Top Med Chem. 2016. PMID: 26585932 Review.
Large-scale High-throughput Screening Revealed 5'-(carbonylamino)-2,3'- bithiophene-4'-carboxylate as Novel Template for Antibacterial Agents.
Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Ayginin AA, Skvortsov DA, Komarova KS, Zagribelnyy BA, Baimiev AK, Shvetc KY, Baimiev AK, Sofronova AA, Machulkin AE, Petrov RA, Zainullina LF, Maximova MA, Zileeva ZR, Vakhitova YV, Bezrukov DS, Puchinina MM, Dontsova OA. Ivanenkov YA, et al. Among authors: aladinskaya av. Curr Drug Discov Technol. 2020;17(5):716-724. doi: 10.2174/1570163816666190603095521. Curr Drug Discov Technol. 2020. PMID: 31161993
Substituted Furanocoumarins as Novel Class of Antibacterial Translation Inhibitors.
Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Ayginin AA, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Skvortsov DA, Komarova KS, Chemeris AV, Zainullina LF, Maximova MA, Zileeva ZR, Vakhitova YV, Baymiev AK, Baymiev AK, Sofronova AA, Machulkin AE, Petrov RA, Bezrukov DS, Puchinina MM, Lukianov DA, Dontsova OA. Ivanenkov YA, et al. Among authors: aladinskaya av. Comb Chem High Throughput Screen. 2019;22(6):400-410. doi: 10.2174/1386207322666190723110539. Comb Chem High Throughput Screen. 2019. PMID: 31573876
2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials.
Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Veselov MS, Ayginin AA, Skvortsov DA, Komarova KS, Sadovnikov SV, Matniyazov R, Sofronova AA, Malyshev AS, Machulkin AE, Petrov RA, Lukianov D, Iarovenko S, Bezrukov DS, Baymiev AK, Dontsova OA. Ivanenkov YA, et al. Among authors: aladinskaya av. J Antibiot (Tokyo). 2019 Nov;72(11):827-833. doi: 10.1038/s41429-019-0211-y. Epub 2019 Jul 29. J Antibiot (Tokyo). 2019. PMID: 31358913
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials.
Veselov MS, Ivanenkov YA, Yamidanov RS, Osterman IA, Sergiev PV, Aladinskiy VA, Aladinskaya AV, Terentiev VA, Ayginin AA, Skvortsov DA, Komarova KS, Chemeris AV, Baimiev AK, Sofronova AA, Machulkin AE, Petrov RA, Maklakova SY, Bezrukov DS, Filkov GI, Zainullina LF, Maximova MA, Zileeva ZR, Kartsev VG, Vakhitova YV, Dontsova OA. Veselov MS, et al. Among authors: aladinskaya av. Mol Divers. 2020 Feb;24(1):233-239. doi: 10.1007/s11030-019-09946-3. Epub 2019 Apr 4. Mol Divers. 2020. PMID: 30949901
16 results