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Probing the Ligand-Binding Pocket of BTN3A1.
J Med Chem. 2019 Jul 25;62(14):6814-6823. doi: 10.1021/acs.jmedchem.9b00825. Epub 2019 Jul 3.
J Med Chem. 2019.
PMID: 31268699
Free PMC article.
Phosphinophosphonates and Their Tris-pivaloyloxymethyl Prodrugs Reveal a Negatively Cooperative Butyrophilin Activation Mechanism.
Shippy RR, Lin X, Agabiti SS, Li J, Zangari BM, Foust BJ, Poe MM, Hsiao CC, Vinogradova O, Wiemer DF, Wiemer AJ.
Shippy RR, et al. Among authors: agabiti ss.
J Med Chem. 2017 Mar 23;60(6):2373-2382. doi: 10.1021/acs.jmedchem.6b00965. Epub 2017 Mar 1.
J Med Chem. 2017.
PMID: 28218845
Free PMC article.
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Toward Broad Spectrum Dihydrofolate Reductase Inhibitors Targeting Trimethoprim Resistant Enzymes Identified in Clinical Isolates of Methicillin Resistant Staphylococcus aureus.
Reeve SM, Si D, Krucinska J, Yan Y, Viswanathan K, Wang S, Holt GT, Frenkel MS, Ojewole AA, Estrada A, Agabiti SS, Alverson JB, Gibson ND, Priestley ND, Wiemer AJ, Donald BR, Wright DL.
Reeve SM, et al. Among authors: agabiti ss.
ACS Infect Dis. 2019 Nov 8;5(11):1896-1906. doi: 10.1021/acsinfecdis.9b00222. Epub 2019 Oct 15.
ACS Infect Dis. 2019.
PMID: 31565920
Free PMC article.
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Molecular mechanisms linking geranylgeranyl diphosphate synthase to cell survival and proliferation.
Agabiti SS, Liang Y, Wiemer AJ.
Agabiti SS, et al.
Mol Membr Biol. 2016 Mar;33(1-2):1-11. doi: 10.1080/09687688.2016.1213432. Epub 2016 Aug 18.
Mol Membr Biol. 2016.
PMID: 27537059
Free PMC article.
Review.
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Geranylgeranyl diphosphate synthase inhibition induces apoptosis that is dependent upon GGPP depletion, ERK phosphorylation and caspase activation.
Agabiti SS, Li J, Wiemer AJ.
Agabiti SS, et al.
Cell Death Dis. 2017 Mar 16;8(3):e2678. doi: 10.1038/cddis.2017.101.
Cell Death Dis. 2017.
PMID: 28300835
Free PMC article.
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Regulation of the Notch-ATM-abl axis by geranylgeranyl diphosphate synthase inhibition.
Agabiti SS, Li J, Dong W, Poe MM, Wiemer AJ.
Agabiti SS, et al.
Cell Death Dis. 2019 Sep 30;10(10):733. doi: 10.1038/s41419-019-1973-7.
Cell Death Dis. 2019.
PMID: 31570763
Free PMC article.
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A genome-wide single-cell 3D genome atlas of lung cancer progression.
Liu M, Jin S, Agabiti SS, Jensen TB, Yang T, Radda JSD, Ruiz CF, Baldissera G, Muzumdar MD, Wang S.
Liu M, et al. Among authors: agabiti ss.
bioRxiv [Preprint]. 2023 Jul 24:2023.07.23.550157. doi: 10.1101/2023.07.23.550157.
bioRxiv. 2023.
PMID: 37546882
Free PMC article.
Preprint.
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