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Active glutaminase C self-assembles into a supratetrameric oligomer that can be disrupted by an allosteric inhibitor.
Ferreira AP, Cassago A, Gonçalves Kde A, Dias MM, Adamoski D, Ascenção CF, Honorato RV, de Oliveira JF, Ferreira IM, Fornezari C, Bettini J, Oliveira PS, Paes Leme AF, Portugal RV, Ambrosio AL, Dias SM. Ferreira AP, et al. Among authors: adamoski d. J Biol Chem. 2013 Sep 27;288(39):28009-20. doi: 10.1074/jbc.M113.501346. Epub 2013 Aug 8. J Biol Chem. 2013. PMID: 23935106 Free PMC article.
Human mitochondrial pyruvate carrier 2 as an autonomous membrane transporter.
Nagampalli RSK, Quesñay JEN, Adamoski D, Islam Z, Birch J, Sebinelli HG, Girard RMBM, Ascenção CFR, Fala AM, Pauletti BA, Consonni SR, de Oliveira JF, Silva ACT, Franchini KG, Leme AFP, Silber AM, Ciancaglini P, Moraes I, Dias SMG, Ambrosio ALB. Nagampalli RSK, et al. Among authors: adamoski d. Sci Rep. 2018 Feb 22;8(1):3510. doi: 10.1038/s41598-018-21740-z. Sci Rep. 2018. PMID: 29472561 Free PMC article.
Dual inhibition of glutaminase and carnitine palmitoyltransferase decreases growth and migration of glutaminase inhibition-resistant triple-negative breast cancer cells.
Reis LMD, Adamoski D, Ornitz Oliveira Souza R, Rodrigues Ascenção CF, Sousa de Oliveira KR, Corrêa-da-Silva F, Malta de Sá Patroni F, Meira Dias M, Consonni SR, Mendes de Moraes-Vieira PM, Silber AM, Dias SMG. Reis LMD, et al. Among authors: adamoski d. J Biol Chem. 2019 Jun 14;294(24):9342-9357. doi: 10.1074/jbc.RA119.008180. Epub 2019 Apr 30. J Biol Chem. 2019. PMID: 31040181 Free PMC article.
GLS2 is protumorigenic in breast cancers.
Dias MM, Adamoski D, Dos Reis LM, Ascenção CFR, de Oliveira KRS, Mafra ACP, da Silva Bastos AC, Quintero M, de G Cassago C, Ferreira IM, Fidelis CHV, Rocco SA, Bajgelman MC, Stine Z, Berindan-Neagoe I, Calin GA, Ambrosio ALB, Dias SMG. Dias MM, et al. Among authors: adamoski d. Oncogene. 2020 Jan;39(3):690-702. doi: 10.1038/s41388-019-1007-z. Epub 2019 Sep 20. Oncogene. 2020. PMID: 31541193
High-Throughput Screening Reveals New Glutaminase Inhibitor Molecules.
E Costa RK, Rodrigues CT, H Campos JC, Paradela LS, Dias MM, Novaes da Silva B, de Valega Negrao CVZ, Gonçalves KA, Ascenção CFR, Adamoski D, Mercaldi GF, Bastos ACS, Batista FAH, Figueira AC, Cordeiro AT, Ambrosio ALB, Guido RVC, Dias SMG. E Costa RK, et al. Among authors: adamoski d. ACS Pharmacol Transl Sci. 2021 Dec 1;4(6):1849-1866. doi: 10.1021/acsptsci.1c00226. eCollection 2021 Dec 10. ACS Pharmacol Transl Sci. 2021. PMID: 34927015 Free PMC article.
Leptin Signaling Suppression in Macrophages Improves Immunometabolic Outcomes in Obesity.
Monteiro LB, Prodonoff JS, Favero de Aguiar C, Correa-da-Silva F, Castoldi A, Bakker NVT, Davanzo GG, Castelucci B, Pereira JADS, Curtis J, Büscher J, Reis LMD, Castro G, Ribeiro G, Virgílio-da-Silva JV, Adamoski D, Dias SMG, Consonni SR, Donato J, Pearce EJ, Câmara NOS, Moraes-Vieira PM. Monteiro LB, et al. Among authors: adamoski d. Diabetes. 2022 Jul 1;71(7):1546-1561. doi: 10.2337/db21-0842. Diabetes. 2022. PMID: 35377454
UV 254 nm is more efficient than UV 222 nm in inactivating SARS-CoV-2 present in human saliva.
Sesti-Costa R, Negrão CVZ, Shimizu JF, Nagai A, Tavares RSN, Adamoski D, Costa W, Fontoura MA, da Silva TJ, de Barros A, Girasole A, de Carvalho M, Teixeira VC, Ambrosio ALB, Granja F, Proença-Módena JL, Marques RE, Dias SMG. Sesti-Costa R, et al. Among authors: adamoski d. Photodiagnosis Photodyn Ther. 2022 Sep;39:103015. doi: 10.1016/j.pdpdt.2022.103015. Epub 2022 Jul 14. Photodiagnosis Photodyn Ther. 2022. PMID: 35843562 Free PMC article.
36 results