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New quinoline derivatives demonstrate a promising antimalarial activity against Plasmodium falciparum in vitro and Plasmodium berghei in vivo.
Soares RR, da Silva JM, Carlos BC, da Fonseca CC, de Souza LS, Lopes FV, de Paula Dias RM, Moreira PO, Abramo C, Viana GH, de Pila Varotti F, da Silva AD, Scopel KK. Soares RR, et al. Among authors: abramo c. Bioorg Med Chem Lett. 2015 Jun 1;25(11):2308-13. doi: 10.1016/j.bmcl.2015.04.014. Epub 2015 Apr 11. Bioorg Med Chem Lett. 2015. PMID: 25920564
Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability.
Guimarães DSM, de Sousa Luz LS, do Nascimento SB, Silva LR, de Miranda Martins NR, de Almeida HG, de Souza Reis V, Maluf SEC, Budu A, Marinho JA, Abramo C, Carmona AK, da Silva MG, da Silva GR, Kemmer VM, Butera AP, Ribeiro-Viana RM, Gazarini ML, Júnior CSN, Guimarães L, Dos Santos FV, de Castro WV, Viana GHR, de Brito CFA, de Pilla Varotti F. Guimarães DSM, et al. Among authors: abramo c. Eur J Pharm Sci. 2019 Oct 1;138:105015. doi: 10.1016/j.ejps.2019.105015. Epub 2019 Jul 22. Eur J Pharm Sci. 2019. PMID: 31344442
In vitro and in vivo antiplasmodial activity of novel quinoline derivative compounds by molecular hybridization.
Marinho JA, Martins Guimarães DS, Glanzmann N, de Almeida Pimentel G, Karine da Costa Nunes I, Gualberto Pereira HM, Navarro M, de Pilla Varotti F, David da Silva A, Abramo C. Marinho JA, et al. Among authors: abramo c. Eur J Med Chem. 2021 Apr 5;215:113271. doi: 10.1016/j.ejmech.2021.113271. Epub 2021 Feb 8. Eur J Med Chem. 2021. PMID: 33596489
Prevalence and risk factors for giardiasis and soil-transmitted helminthiasis in three municipalities of Southeastern Minas Gerais State, Brazil: risk factors for giardiasis and soil-transmitted helminthiasis.
Pinheiro Ide O, de Castro MF, Mitterofhe A, Pires FA, Abramo C, Ribeiro LC, Tibiriçá SH, Coimbra ES. Pinheiro Ide O, et al. Among authors: abramo c. Parasitol Res. 2011 May;108(5):1123-30. doi: 10.1007/s00436-010-2154-x. Epub 2011 Jan 18. Parasitol Res. 2011. PMID: 21243507
56 results