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Interindividual Variability in Cytochrome P450 3A and 1A Activity Influences Sunitinib Metabolism and Bioactivation.
Chem Res Toxicol. 2022 May 16;35(5):792-806. doi: 10.1021/acs.chemrestox.1c00426. Epub 2022 Apr 28.
Chem Res Toxicol. 2022.
PMID: 35484684
Free PMC article.
Cytochromes P450 1A2 and 3A4 Catalyze the Metabolic Activation of Sunitinib.
Amaya GM, Durandis R, Bourgeois DS, Perkins JA, Abouda AA, Wines KJ, Mohamud M, Starks SA, Daniels RN, Jackson KD.
Amaya GM, et al. Among authors: abouda aa.
Chem Res Toxicol. 2018 Jul 16;31(7):570-584. doi: 10.1021/acs.chemrestox.8b00005. Epub 2018 Jun 18.
Chem Res Toxicol. 2018.
PMID: 29847931
Free PMC article.
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Interindividual Variation in CYP3A Activity Influences Lapatinib Bioactivation.
Bissada JE, Truong V, Abouda AA, Wines KJ, Crouch RD, Jackson KD.
Bissada JE, et al. Among authors: abouda aa.
Drug Metab Dispos. 2019 Nov;47(11):1257-1269. doi: 10.1124/dmd.119.088823. Epub 2019 Sep 6.
Drug Metab Dispos. 2019.
PMID: 31492693
Free PMC article.
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Detoxication versus Bioactivation Pathways of Lapatinib In Vitro: UGT1A1 Catalyzes the Hepatic Glucuronidation of Debenzylated Lapatinib.
Nardone-White DT, Bissada JE, Abouda AA, Jackson KD.
Nardone-White DT, et al. Among authors: abouda aa.
Drug Metab Dispos. 2021 Mar;49(3):233-244. doi: 10.1124/dmd.120.000236. Epub 2020 Dec 29.
Drug Metab Dispos. 2021.
PMID: 33376146
Free PMC article.
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