Abdelgawad MA - Search Results

1

Piperidine: A Versatile Heterocyclic Ring for Developing Monoamine Oxidase Inhibitors.

Jayan J, Chandran N, Thekkantavida AC, Abdelgawad MA, Ghoneim MM, Shaker ME, Uniyal P, Benny F, Zachariah SM, Kumar S, Kim H, Mathew B. Jayan J, et al. Among authors: abdelgawad ma. ACS Omega. 2023 Oct 3;8(41):37731-37751. doi: 10.1021/acsomega.3c05883. eCollection 2023 Oct 17. ACS Omega. 2023. PMID: 37867639 Free PMC article. Review.

2

Design, Synthesis and Biological Evaluation of New HDAC1 and HDAC2 Inhibitors Endowed with Ligustrazine as a Novel Cap Moiety.

Al-Sanea MM, Gotina L, Mohamed MF, Grace Thomas Parambi D, Gomaa HAM, Mathew B, Youssif BGM, Alharbi KS, Elsayed ZM, Abdelgawad MA, Eldehna WM. Al-Sanea MM, et al. Among authors: abdelgawad ma. Drug Des Devel Ther. 2020 Feb 4;14:497-508. doi: 10.2147/DDDT.S237957. eCollection 2020. Drug Des Devel Ther. 2020. PMID: 32103894 Free PMC article.

3

Revealing the role of fluorine pharmacophore in chalcone scaffold for shifting the MAO-B selectivity: investigation of a detailed molecular dynamics and quantum chemical study.

Olotu FA, Joy M, Abdelgawad MA, Narayanan SE, Soliman ME, Mathew B. Olotu FA, et al. Among authors: abdelgawad ma. J Biomol Struct Dyn. 2021 Oct;39(16):6126-6139. doi: 10.1080/07391102.2020.1796803. Epub 2020 Jul 24. J Biomol Struct Dyn. 2021. PMID: 32705963

4

Design, Synthesis, and Biological Evaluation of Pyridazinones Containing the (2-Fluorophenyl) Piperazine Moiety as Selective MAO-B Inhibitors.

Çeçen M, Oh JM, Özdemir Z, Büyüktuncel SE, Uysal M, Abdelgawad MA, Musa A, Gambacorta N, Nicolotti O, Mathew B, Kim H. Çeçen M, et al. Among authors: abdelgawad ma. Molecules. 2020 Nov 17;25(22):5371. doi: 10.3390/molecules25225371. Molecules. 2020. PMID: 33212876 Free PMC article.

5

Morpholine-based chalcones as dual-acting monoamine oxidase-B and acetylcholinesterase inhibitors: synthesis and biochemical investigations.

Sasidharan R, Eom BH, Heo JH, Park JE, Abdelgawad MA, Musa A, Gambacorta N, Nicolotti O, Manju SL, Mathew B, Kim H. Sasidharan R, et al. Among authors: abdelgawad ma. J Enzyme Inhib Med Chem. 2021 Dec;36(1):188-197. doi: 10.1080/14756366.2020.1842390. J Enzyme Inhib Med Chem. 2021. PMID: 33430657 Free PMC article.

6

A New CDK2 Inhibitor with 3-Hydrazonoindolin-2-One Scaffold Endowed with Anti-Breast Cancer Activity: Design, Synthesis, Biological Evaluation, and In Silico Insights.

Al-Sanea MM, Obaidullah AJ, Shaker ME, Chilingaryan G, Alanazi MM, Alsaif NA, Alkahtani HM, Alsubaie SA, Abdelgawad MA. Al-Sanea MM, et al. Among authors: abdelgawad ma. Molecules. 2021 Jan 14;26(2):412. doi: 10.3390/molecules26020412. Molecules. 2021. PMID: 33466812 Free PMC article.

7

Development of Halogenated Pyrazolines as Selective Monoamine Oxidase-B Inhibitors: Deciphering via Molecular Dynamics Approach.

Nair AS, Oh JM, Koyiparambath VP, Kumar S, Sudevan ST, Soremekun O, Soliman ME, Khames A, Abdelgawad MA, Pappachen LK, Mathew B, Kim H. Nair AS, et al. Among authors: abdelgawad ma. Molecules. 2021 May 28;26(11):3264. doi: 10.3390/molecules26113264. Molecules. 2021. PMID: 34071665 Free PMC article.

8

Novel Phenolic Compounds as Potential Dual EGFR and COX-2 Inhibitors: Design, Semisynthesis, in vitro Biological Evaluation and in silico Insights.

Abdelgawad MA, Musa A, Almalki AH, Alzarea SI, Mostafa EM, Hegazy MM, Mostafa-Hedeab G, Ghoneim MM, Parambi DGT, Bakr RB, Al-Muaikel NS, Alanazi AS, Alharbi M, Ahmad W, Bukhari SNA, Al-Sanea MM. Abdelgawad MA, et al. Drug Des Devel Ther. 2021 May 31;15:2325-2337. doi: 10.2147/DDDT.S310820. eCollection 2021. Drug Des Devel Ther. 2021. PMID: 34103896 Free PMC article.

9

Trimethoxylated Halogenated Chalcones as Dual Inhibitors of MAO-B and BACE-1 for the Treatment of Neurodegenerative Disorders.

Vishal PK, Oh JM, Khames A, Abdelgawad MA, Nair AS, Nath LR, Gambacorta N, Ciriaco F, Nicolotti O, Kim H, Mathew B. Vishal PK, et al. Among authors: abdelgawad ma. Pharmaceutics. 2021 Jun 8;13(6):850. doi: 10.3390/pharmaceutics13060850. Pharmaceutics. 2021. PMID: 34201128 Free PMC article.

10

Strawberry and Ginger Silver Nanoparticles as Potential Inhibitors for SARS-CoV-2 Assisted by In Silico Modeling and Metabolic Profiling.

Al-Sanea MM, Abelyan N, Abdelgawad MA, Musa A, Ghoneim MM, Al-Warhi T, Aljaeed N, Alotaibi OJ, Alnusaire TS, Abdelwahab SF, Helmy A, Abdelmohsen UR, Youssif KA. Al-Sanea MM, et al. Among authors: abdelgawad ma. Antibiotics (Basel). 2021 Jul 6;10(7):824. doi: 10.3390/antibiotics10070824. Antibiotics (Basel). 2021. PMID: 34356745 Free PMC article.

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