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Encorafenib Acts as a Dual-Activity Chemosensitizer through Its Inhibitory Effect on ABCC1 Transporter In Vitro and Ex Vivo.
Pharmaceutics. 2022 Nov 24;14(12):2595. doi: 10.3390/pharmaceutics14122595.
Pharmaceutics. 2022.
PMID: 36559089
Free PMC article.
Tepotinib Inhibits Several Drug Efflux Transporters and Biotransformation Enzymes: The Role in Drug-Drug Interactions and Targeting Cytostatic Resistance In Vitro and Ex Vivo.
Vagiannis D, Budagaga Y, Morell A, Zhang Y, Novotná E, Skarka A, Kammerer S, Küpper JH, Hanke I, Rozkoš T, Hofman J.
Vagiannis D, et al.
Int J Mol Sci. 2021 Nov 3;22(21):11936. doi: 10.3390/ijms222111936.
Int J Mol Sci. 2021.
PMID: 34769363
Free PMC article.
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