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High amount of lecithin facilitates oral delivery of a poorly soluble pyrazoloquinolinone ligand formulated in lipid nanoparticles: Physicochemical, structural and pharmacokinetic performances.
Int J Pharm. 2023 Feb 25;633:122613. doi: 10.1016/j.ijpharm.2023.122613. Epub 2023 Jan 16.
Int J Pharm. 2023.
PMID: 36657554
Free PMC article.
Nanocrystal dispersion of DK-I-56-1, a poorly soluble pyrazoloquinolinone positive modulator of α6 GABAA receptors: Formulation approach toward improved in vivo performance.
Mitrović JR, Divović B, Knutson DE, Đoković JB, Vulić PJ, Randjelović DV, Dobričić VD, Čalija BR, Cook JM, Savić MM, Savić SD.
Mitrović JR, et al. Among authors: dokovic jb.
Eur J Pharm Sci. 2020 Sep 1;152:105432. doi: 10.1016/j.ejps.2020.105432. Epub 2020 Jun 18.
Eur J Pharm Sci. 2020.
PMID: 32565331
Free PMC article.
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Curcumin Loaded PEGylated Nanoemulsions Designed for Maintained Antioxidant Effects and Improved Bioavailability: A Pilot Study on Rats.
Đoković JB, Savić SM, Mitrović JR, Nikolic I, Marković BD, Randjelović DV, Antic-Stankovic J, Božić D, Cekić ND, Stevanović V, Batinić B, Aranđelović J, Savić MM, Savić SD.
Đoković JB, et al.
Int J Mol Sci. 2021 Jul 27;22(15):7991. doi: 10.3390/ijms22157991.
Int J Mol Sci. 2021.
PMID: 34360758
Free PMC article.
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Overcoming the Low Oral Bioavailability of Deuterated Pyrazoloquinolinone Ligand DK-I-60-3 by Nanonization: A Knowledge-Based Approach.
Mitrović JR, Divović-Matović B, Knutson DE, Đoković JB, Kremenović A, Dobričić VD, Randjelović DV, Pantelić I, Cook JM, Savić MM, Savić SD.
Mitrović JR, et al. Among authors: dokovic jb.
Pharmaceutics. 2021 Jul 31;13(8):1188. doi: 10.3390/pharmaceutics13081188.
Pharmaceutics. 2021.
PMID: 34452149
Free PMC article.
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The Impact of the Oil Phase Selection on Physicochemical Properties, Long-Term Stability, In Vitro Performance and Injectability of Curcumin-Loaded PEGylated Nanoemulsions.
Đoković JB, Demisli S, Savić SM, Marković BD, Cekić ND, Randjelovic DV, Mitrović JR, Lunter DJ, Papadimitriou V, Xenakis A, Savić SD.
Đoković JB, et al.
Pharmaceutics. 2022 Aug 10;14(8):1666. doi: 10.3390/pharmaceutics14081666.
Pharmaceutics. 2022.
PMID: 36015291
Free PMC article.
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Parenteral Lipid-Based Nanoparticles for CNS Disorders: Integrating Various Facets of Preclinical Evaluation towards More Effective Clinical Translation.
Ilić T, Đoković JB, Nikolić I, Mitrović JR, Pantelić I, Savić SD, Savić MM.
Ilić T, et al. Among authors: dokovic jb.
Pharmaceutics. 2023 Jan 29;15(2):443. doi: 10.3390/pharmaceutics15020443.
Pharmaceutics. 2023.
PMID: 36839768
Free PMC article.
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