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Year | Number of Results |
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2008 | 1 |
2009 | 1 |
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Modifications of human carboxylesterase for improved prodrug activation.
Expert Opin Drug Metab Toxicol. 2008 Sep;4(9):1153-65. doi: 10.1517/17425255.4.9.1153.
Expert Opin Drug Metab Toxicol. 2008.
PMID: 18721110
Free PMC article.
Review.
Requirements for mammalian carboxylesterase inhibition by substituted ethane-1,2-diones.
Parkinson EI, Jason Hatfield M, Tsurkan L, Hyatt JL, Edwards CC, Hicks LD, Yan B, Potter PM.
Parkinson EI, et al.
Bioorg Med Chem. 2011 Aug 1;19(15):4635-43. doi: 10.1016/j.bmc.2011.06.012. Epub 2011 Jul 4.
Bioorg Med Chem. 2011.
PMID: 21733699
Free PMC article.
Item in Clipboard
Organ-specific carboxylesterase profiling identifies the small intestine and kidney as major contributors of activation of the anticancer prodrug CPT-11.
Hatfield MJ, Tsurkan L, Garrett M, Shaver TM, Hyatt JL, Edwards CC, Hicks LD, Potter PM.
Hatfield MJ, et al.
Biochem Pharmacol. 2011 Jan 1;81(1):24-31. doi: 10.1016/j.bcp.2010.09.001. Epub 2010 Sep 15.
Biochem Pharmacol. 2011.
PMID: 20833148
Free PMC article.
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Improved, selective, human intestinal carboxylesterase inhibitors designed to modulate 7-ethyl-10-[4-(1-piperidino)-1-piperidino]carbonyloxycamptothecin (Irinotecan; CPT-11) toxicity.
Hicks LD, Hyatt JL, Stoddard S, Tsurkan L, Edwards CC, Wadkins RM, Potter PM.
Hicks LD, et al.
J Med Chem. 2009 Jun 25;52(12):3742-52. doi: 10.1021/jm9001296.
J Med Chem. 2009.
PMID: 19534556
Free PMC article.
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