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Metabolite Identification of HIV-1 Capsid Modulators PF74 and 11L in Human Liver Microsomes.
Metabolites. 2022 Aug 16;12(8):752. doi: 10.3390/metabo12080752.
Metabolites. 2022.
PMID: 36005624
Free PMC article.
Discovery of low-molecular-weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability.
Jiang X, Gao Z, Sharma PP, Kumar S, Rathi B, Ji X, Dai J, Xie M, Dong G, Xu S, De Clercq E, Pannecouque C, Dick A, Zhan P, Liu X.
Jiang X, et al.
J Med Virol. 2024 Apr;96(4):e29594. doi: 10.1002/jmv.29594.
J Med Virol. 2024.
PMID: 38576317
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