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3-Arylidene-2-oxindoles as GSK3β inhibitors and anti-thrombotic agents.
Babkov D, Bezsonova E, Sirotenko V, Othman E, Klochkov V, Sosonyuk S, Lozinskaya N, Spasov A. Babkov D, et al. Among authors: klochkov v. Bioorg Med Chem Lett. 2023 May 1;87:129283. doi: 10.1016/j.bmcl.2023.129283. Epub 2023 Apr 11. Bioorg Med Chem Lett. 2023. PMID: 37054760 Free PMC article.
3-Arylidene-2-oxindoles as Potent NRH:Quinone Oxidoreductase 2 Inhibitors.
Lozinskaya NA, Bezsonova EN, Dubar M, Melekhina DD, Bazanov DR, Bunev AS, Grigor'eva OB, Klochkov VG, Sokolova EV, Babkov DA, Spasov AA, Sosonyuk SE. Lozinskaya NA, et al. Among authors: klochkov vg. Molecules. 2023 Jan 25;28(3):1174. doi: 10.3390/molecules28031174. Molecules. 2023. PMID: 36770840 Free PMC article.
Guanidine Derivatives of Quinazoline-2,4(1H,3H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents.
Spasov A, Ozerov A, Kosolapov V, Gurova N, Kucheryavenko A, Naumenko L, Babkov D, Sirotenko V, Taran A, Borisov A, Sokolova E, Klochkov V, Merezhkina D, Miroshnikov M, Ovsyankina N, Smirnov A, Velikorodnaya Y. Spasov A, et al. Among authors: klochkov v. Life (Basel). 2022 Oct 20;12(10):1647. doi: 10.3390/life12101647. Life (Basel). 2022. PMID: 36295082 Free PMC article.
Synthesis and multifaceted pharmacological activity of novel quinazoline NHE-1 inhibitors.
Spasov A, Ozerov A, Vassiliev P, Kosolapov V, Gurova N, Kucheryavenko A, Naumenko L, Babkov D, Sirotenko V, Taran A, Litvinov R, Borisov A, Klochkov V, Merezhkina D, Miroshnikov M, Uskov G, Ovsyankina N. Spasov A, et al. Among authors: klochkov v. Sci Rep. 2021 Dec 21;11(1):24380. doi: 10.1038/s41598-021-03722-w. Sci Rep. 2021. PMID: 34934125 Free PMC article.
Discovery of Nitro-azolo[1,5-a]pyrimidines with Anti-Inflammatory and Protective Activity against LPS-Induced Acute Lung Injury.
Spasov A, Kosolapov V, Babkov D, Klochkov V, Sokolova E, Miroshnikov M, Borisov A, Velikorodnaya Y, Smirnov A, Savateev K, Fedotov V, Kotovskaya S, Rusinov V. Spasov A, et al. Among authors: klochkov v. Pharmaceuticals (Basel). 2022 Apr 27;15(5):537. doi: 10.3390/ph15050537. Pharmaceuticals (Basel). 2022. PMID: 35631365 Free PMC article.