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Development of a Potent Nurr1 Agonist Tool for In Vivo Applications.
J Med Chem. 2023 May 11;66(9):6391-6402. doi: 10.1021/acs.jmedchem.3c00415. Epub 2023 Apr 26.
J Med Chem. 2023.
PMID: 37127285
Free PMC article.
Exploring Fatty Acid Mimetics as NR4A Ligands.
Stiller T, Merk D.
Stiller T, et al.
J Med Chem. 2023 Nov 23;66(22):15362-15369. doi: 10.1021/acs.jmedchem.3c01467. Epub 2023 Nov 2.
J Med Chem. 2023.
PMID: 37918435
Free PMC article.
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De Novo Design of Nurr1 Agonists via Fragment-Augmented Generative Deep Learning in Low-Data Regime.
Ballarotto M, Willems S, Stiller T, Nawa F, Marschner JA, Grisoni F, Merk D.
Ballarotto M, et al. Among authors: stiller t.
J Med Chem. 2023 Jun 22;66(12):8170-8177. doi: 10.1021/acs.jmedchem.3c00485. Epub 2023 May 31.
J Med Chem. 2023.
PMID: 37256819
Free PMC article.
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