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2018 3
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Page 1
Strategies for Delivery of siRNAs to Ovarian Cancer Cells.
Farra R, Maruna M, Perrone F, Grassi M, Benedetti F, Maddaloni M, El Boustani M, Parisi S, Rizzolio F, Forte G, Zanconati F, Cemazar M, Kamensek U, Dapas B, Grassi G. Farra R, et al. Among authors: el boustani m. Pharmaceutics. 2019 Oct 22;11(10):547. doi: 10.3390/pharmaceutics11100547. Pharmaceutics. 2019. PMID: 31652539 Free PMC article. Review.
Polymer-Mediated Delivery of siRNAs to Hepatocellular Carcinoma: Variables Affecting Specificity and Effectiveness.
Farra R, Musiani F, Perrone F, Čemažar M, Kamenšek U, Tonon F, Abrami M, Ručigaj A, Grassi M, Pozzato G, Bonazza D, Zanconati F, Forte G, El Boustani M, Scarabel L, Garziera M, Russo Spena C, De Stefano L, Salis B, Toffoli G, Rizzolio F, Grassi G, Dapas B. Farra R, et al. Among authors: el boustani m. Molecules. 2018 Mar 28;23(4):777. doi: 10.3390/molecules23040777. Molecules. 2018. PMID: 29597300 Free PMC article. Review.
A Guide to PIN1 Function and Mutations Across Cancers.
El Boustani M, De Stefano L, Caligiuri I, Mouawad N, Granchi C, Canzonieri V, Tuccinardi T, Giordano A, Rizzolio F. El Boustani M, et al. Front Pharmacol. 2019 Jan 22;9:1477. doi: 10.3389/fphar.2018.01477. eCollection 2018. Front Pharmacol. 2019. PMID: 30723410 Free PMC article.
Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors.
Bononi G, Granchi C, Lapillo M, Giannotti M, Nieri D, Fortunato S, Boustani ME, Caligiuri I, Poli G, Carlson KE, Kim SH, Macchia M, Martinelli A, Rizzolio F, Chicca A, Katzenellenbogen JA, Minutolo F, Tuccinardi T. Bononi G, et al. Among authors: boustani me. Eur J Med Chem. 2018 Sep 5;157:817-836. doi: 10.1016/j.ejmech.2018.08.038. Epub 2018 Aug 16. Eur J Med Chem. 2018. PMID: 30144699
Virtual screening identifies a PIN1 inhibitor with possible antiovarian cancer effects.
Russo Spena C, De Stefano L, Poli G, Granchi C, El Boustani M, Ecca F, Grassi G, Grassi M, Canzonieri V, Giordano A, Tuccinardi T, Caligiuri I, Rizzolio F. Russo Spena C, et al. Among authors: el boustani m. J Cell Physiol. 2019 Sep;234(9):15708-15716. doi: 10.1002/jcp.28224. Epub 2019 Jan 29. J Cell Physiol. 2019. PMID: 30697729
Optimization of a Benzoylpiperidine Class Identifies a Highly Potent and Selective Reversible Monoacylglycerol Lipase (MAGL) Inhibitor.
Granchi C, Lapillo M, Glasmacher S, Bononi G, Licari C, Poli G, El Boustani M, Caligiuri I, Rizzolio F, Gertsch J, Macchia M, Minutolo F, Tuccinardi T, Chicca A. Granchi C, et al. Among authors: el boustani m. J Med Chem. 2019 Feb 28;62(4):1932-1958. doi: 10.1021/acs.jmedchem.8b01483. Epub 2019 Feb 11. J Med Chem. 2019. PMID: 30715876