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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2007 1
2012 1
2013 1
2014 1
2015 1
2016 3
2017 2
2018 6
2019 2
2020 2
2021 3
2022 2
2023 1
2024 0

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24 results

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Page 1
3-hydroxy-L-kynurenamine is an immunomodulatory biogenic amine.
Clement CC, D'Alessandro A, Thangaswamy S, Chalmers S, Furtado R, Spada S, Mondanelli G, Ianni F, Gehrke S, Gargaro M, Manni G, Cara LCL, Runge P, Tsai WL, Karaman S, Arasa J, Fernandez-Rodriguez R, Beck A, Macchiarulo A, Gadina M, Halin C, Fallarino F, Skobe M, Veldhoen M, Moretti S, Formenti S, Demaria S, Soni RK, Galarini R, Sardella R, Lauvau G, Putterman C, Alitalo K, Grohmann U, Santambrogio L. Clement CC, et al. Among authors: cara lcl. Nat Commun. 2021 Jul 21;12(1):4447. doi: 10.1038/s41467-021-24785-3. Nat Commun. 2021. PMID: 34290243 Free PMC article.
1,2-Diphenoxiethane salts as potent antiplasmodial agents.
Schiafino-Ortega S, Baglioni E, Pérez-Moreno G, Marco PR, Marco C, González-Pacanowska D, Ruiz-Pérez LM, Carrasco-Jiménez MP, López-Cara LC. Schiafino-Ortega S, et al. Among authors: lopez cara lc. Bioorg Med Chem Lett. 2018 Aug 1;28(14):2485-2489. doi: 10.1016/j.bmcl.2018.05.060. Epub 2018 May 31. Bioorg Med Chem Lett. 2018. PMID: 29880399
New non-symmetrical choline kinase inhibitors.
Schiaffino-Ortega S, López-Cara LC, Ríos-Marco P, Carrasco-Jimenez MP, Gallo MA, Espinosa A, Marco C, Entrena A. Schiaffino-Ortega S, et al. Among authors: lopez cara lc. Bioorg Med Chem. 2013 Nov 15;21(22):7146-54. doi: 10.1016/j.bmc.2013.09.003. Epub 2013 Sep 11. Bioorg Med Chem. 2013. PMID: 24080101
New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action.
Luque-Navarro PM, Carrasco-Jiménez MP, Goracci L, Paredes JM, Espinar-Barranco L, Valverde-Pozo J, Torretta A, Parisini E, Mariotto E, Marchioro C, Laso A, Marco C, Viola G, Lanari D, López Cara LC. Luque-Navarro PM, et al. Among authors: lopez cara lc. Eur J Med Chem. 2023 Jan 15;246:115003. doi: 10.1016/j.ejmech.2022.115003. Epub 2022 Dec 5. Eur J Med Chem. 2023. PMID: 36493617
Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors.
Luque-Navarro PM, Mariotto E, Ballarotto M, Rubbini G, Aguilar-Troyano FJ, Fasiolo A, Torretta A, Parisini E, Macchiarulo A, Laso A, Marco C, Viola G, Carrasco-Jimenez MP, López-Cara LC. Luque-Navarro PM, et al. Among authors: lopez cara lc. Pharmaceutics. 2022 Mar 27;14(4):715. doi: 10.3390/pharmaceutics14040715. Pharmaceutics. 2022. PMID: 35456549 Free PMC article.
Anticancer and Structure Activity Relationship of Non-Symmetrical Choline Kinase Inhibitors.
Schiaffino-Ortega S, Mariotto E, Luque-Navarro PM, Kimatrai-Salvador M, Rios-Marco P, Hurtado-Guerrero R, Marco C, Carrasco-Jimenez MP, Viola G, López-Cara LC. Schiaffino-Ortega S, et al. Among authors: lopez cara lc. Pharmaceutics. 2021 Aug 29;13(9):1360. doi: 10.3390/pharmaceutics13091360. Pharmaceutics. 2021. PMID: 34575436 Free PMC article.
New Compounds with Bioisosteric Replacement of Classic Choline Kinase Inhibitors Show Potent Antiplasmodial Activity.
Aguilar-Troyano FJ, Torretta A, Rubbini G, Fasiolo A, Luque-Navarro PM, Carrasco-Jimenez MP, Pérez-Moreno G, Bosch-Navarrete C, González-Pacanowska D, Parisini E, Lopez-Cara LC. Aguilar-Troyano FJ, et al. Among authors: lopez cara lc. Pharmaceutics. 2021 Nov 2;13(11):1842. doi: 10.3390/pharmaceutics13111842. Pharmaceutics. 2021. PMID: 34834257 Free PMC article.
Lead optimization-hit expansion of new asymmetrical pyridinium/quinolinium compounds as choline kinase α1 inhibitors.
Rubbini G, Buades-Martín AB, Kimatrai-Salvador M, Entrena A, Gallo-Mezo MÁ, Ríos-Marco P, Marco C, Mattiuzzo E, Bortolozzi R, Mariotto E, Greco FA, Macchiarulo A, Carrasco-Jiménez MP, Viola G, López-Cara LC. Rubbini G, et al. Among authors: lopez cara lc. Future Med Chem. 2018 Aug 1;10(15):1769-1786. doi: 10.4155/fmc-2018-0059. Epub 2018 Jul 25. Future Med Chem. 2018. PMID: 30043647
24 results