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Page 1
Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors.
Brem J, Panduwawala T, Hansen JU, Hewitt J, Liepins E, Donets P, Espina L, Farley AJM, Shubin K, Campillos GG, Kiuru P, Shishodia S, Krahn D, Leśniak RK, Schmidt Adrian J, Calvopiña K, Turrientes MC, Kavanagh ME, Lubriks D, Hinchliffe P, Langley GW, Aboklaish AF, Eneroth A, Backlund M, Baran AG, Nielsen EI, Speake M, Kuka J, Robinson J, Grinberga S, Robinson L, McDonough MA, Rydzik AM, Leissing TM, Jimenez-Castellanos JC, Avison MB, Da Silva Pinto S, Pannifer AD, Martjuga M, Widlake E, Priede M, Hopkins Navratilova I, Gniadkowski M, Belfrage AK, Brandt P, Yli-Kauhaluoma J, Bacque E, Page MGP, Björkling F, Tyrrell JM, Spencer J, Lang PA, Baranczewski P, Cantón R, McElroy SP, Jones PS, Baquero F, Suna E, Morrison A, Walsh TR, Schofield CJ. Brem J, et al. Among authors: shubin k. Nat Chem. 2022 Jan;14(1):15-24. doi: 10.1038/s41557-021-00831-x. Epub 2021 Dec 13. Nat Chem. 2022. PMID: 34903857
PLBD: protein-ligand binding database of thermodynamic and kinetic intrinsic parameters.
Lingė D, Gedgaudas M, Merkys A, Petrauskas V, Vaitkus A, Grybauskas A, Paketurytė V, Zubrienė A, Zakšauskas A, Mickevičiūtė A, Smirnovienė J, Baranauskienė L, Čapkauskaitė E, Dudutienė V, Urniežius E, Konovalovas A, Kazlauskas E, Shubin K, Schiöth HB, Chen WY, Ladbury JE, Gražulis S, Matulis D. Lingė D, et al. Among authors: shubin k. Database (Oxford). 2023 Jun 8;2023:baad040. doi: 10.1093/database/baad040. Database (Oxford). 2023. PMID: 37290059 Free PMC article.
Stereodivergent Synthesis of Pseudotabersonine Alkaloids.
Kazak M, Priede M, Shubin K, Bartrum HE, Poisson JF, Suna E. Kazak M, et al. Among authors: shubin k. Org Lett. 2017 Oct 6;19(19):5356-5359. doi: 10.1021/acs.orglett.7b02635. Epub 2017 Sep 13. Org Lett. 2017. PMID: 28901770
Picomolar fluorescent probes for compound affinity determination to carbonic anhydrase IX expressed in live cancer cells.
Matulienė J, Žvinys G, Petrauskas V, Kvietkauskaitė A, Zakšauskas A, Shubin K, Zubrienė A, Baranauskienė L, Kačenauskaitė L, Kopanchuk S, Veiksina S, Paketurytė-Latvė V, Smirnovienė J, Juozapaitienė V, Mickevičiūtė A, Michailovienė V, Jachno J, Stravinskienė D, Sližienė A, Petrošiūtė A, Becker HM, Kazokaitė-Adomaitienė J, Yaromina A, Čapkauskaitė E, Rinken A, Dudutienė V, Dubois LJ, Matulis D. Matulienė J, et al. Among authors: shubin k. Sci Rep. 2022 Oct 21;12(1):17644. doi: 10.1038/s41598-022-22436-1. Sci Rep. 2022. PMID: 36271018 Free PMC article.
Structure-activity relationship studies on the inhibition of the bacterial translation of novel Odilorhabdins analogues.
Loza E, Sarciaux M, Ikaunieks M, Katkevics M, Kukosha T, Trufilkina N, Ryabova V, Shubin K, Pantel L, Serri M, Huseby DL, Cao S, Yadav K, Hjort K, Hughes D, Gualtieri M, Suna E, Racine E. Loza E, et al. Among authors: shubin k. Bioorg Med Chem. 2020 Jun 1;28(11):115469. doi: 10.1016/j.bmc.2020.115469. Epub 2020 Apr 3. Bioorg Med Chem. 2020. PMID: 32279921
11 results