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Page 1
CTP promotes efficient ParB-dependent DNA condensation by facilitating one-dimensional diffusion from parS.
Elife. 2021 Jul 12;10:e67554. doi: 10.7554/eLife.67554.
Elife. 2021.
PMID: 34250901
Free PMC article.
Synthesis of Thicolchicine-Based Conjugates: Investigation towards Bivalent Tubulin/Microtubules Binders.
Bonandi E, Foschi F, Marucci C, Dapiaggi F, Sironi M, Pieraccini S, Christodoulou MS, de Asís Balaguer F, Díaz JF, Zidar N, Passarella D.
Bonandi E, et al. Among authors: de asis balaguer f.
Chempluschem. 2019 Jan;84(1):98-102. doi: 10.1002/cplu.201800497.
Chempluschem. 2019.
PMID: 31950734
Free article.
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Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands.
Balaguer FA, Mühlethaler T, Estévez-Gallego J, Calvo E, Giménez-Abián JF, Risinger AL, Sorensen EJ, Vanderwal CD, Altmann KH, Mooberry SL, Steinmetz MO, Oliva MÁ, Prota AE, Díaz JF.
Balaguer FA, et al.
Int J Mol Sci. 2019 Mar 20;20(6):1392. doi: 10.3390/ijms20061392.
Int J Mol Sci. 2019.
PMID: 30897704
Free PMC article.
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Structure-activity relationships, biological evaluation and structural studies of novel pyrrolonaphthoxazepines as antitumor agents.
Brindisi M, Ulivieri C, Alfano G, Gemma S, de Asís Balaguer F, Khan T, Grillo A, Chemi G, Menchon G, Prota AE, Olieric N, Lucena-Agell D, Barasoain I, Diaz JF, Nebbioso A, Conte M, Lopresti L, Magnano S, Amet R, Kinsella P, Zisterer DM, Ibrahim O, O'Sullivan J, Morbidelli L, Spaccapelo R, Baldari C, Butini S, Novellino E, Campiani G, Altucci L, Steinmetz MO, Brogi S.
Brindisi M, et al. Among authors: de asis balaguer f.
Eur J Med Chem. 2019 Jan 15;162:290-320. doi: 10.1016/j.ejmech.2018.11.004. Epub 2018 Nov 3.
Eur J Med Chem. 2019.
PMID: 30448418
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Triazolopyrimidines Are Microtubule-Stabilizing Agents that Bind the Vinca Inhibitor Site of Tubulin.
Sáez-Calvo G, Sharma A, Balaguer FA, Barasoain I, Rodríguez-Salarichs J, Olieric N, Muñoz-Hernández H, Berbís MÁ, Wendeborn S, Peñalva MA, Matesanz R, Canales Á, Prota AE, Jímenez-Barbero J, Andreu JM, Lamberth C, Steinmetz MO, Díaz JF.
Sáez-Calvo G, et al. Among authors: balaguer fa.
Cell Chem Biol. 2017 Jun 22;24(6):737-750.e6. doi: 10.1016/j.chembiol.2017.05.016. Epub 2017 Jun 1.
Cell Chem Biol. 2017.
PMID: 28579361
Free article.
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Quinolin-6-Yloxyacetamides Are Microtubule Destabilizing Agents That Bind to the Colchicine Site of Tubulin.
Sharma A, Sáez-Calvo G, Olieric N, de Asís Balaguer F, Barasoain I, Lamberth C, Díaz JF, Steinmetz MO.
Sharma A, et al. Among authors: de asis balaguer f.
Int J Mol Sci. 2017 Jun 22;18(7):1336. doi: 10.3390/ijms18071336.
Int J Mol Sci. 2017.
PMID: 28640209
Free PMC article.
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