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Identification of unprecedented ATP-competitive choline kinase inhibitors.
Quartieri F, Nesi M, Avanzi NR, Borghi D, Casale E, Corti E, Cucchi U, Donati D, Fasolini M, Felder ER, Galvani A, Giorgini ML, Lomolino A, Menichincheri M, Orrenius C, Perrera C, Re Depaolini S, Riccardi-Sirtori F, Salsi E, Isacchi A, Gnocchi P. Quartieri F, et al. Bioorg Med Chem Lett. 2021 Nov 1;51:128310. doi: 10.1016/j.bmcl.2021.128310. Epub 2021 Aug 18. Bioorg Med Chem Lett. 2021. PMID: 34416377
A submarine journey: the pyrrole-imidazole alkaloids.
Forte B, Malgesini B, Piutti C, Quartieri F, Scolaro A, Papeo G. Forte B, et al. Among authors: quartieri f. Mar Drugs. 2009 Nov 27;7(4):705-53. doi: 10.3390/md7040705. Mar Drugs. 2009. PMID: 20098608 Free PMC article. Review.
Identification of N,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide (PHA-848125), a potent, orally available cyclin dependent kinase inhibitor.
Brasca MG, Amboldi N, Ballinari D, Cameron A, Casale E, Cervi G, Colombo M, Colotta F, Croci V, D'Alessio R, Fiorentini F, Isacchi A, Mercurio C, Moretti W, Panzeri A, Pastori W, Pevarello P, Quartieri F, Roletto F, Traquandi G, Vianello P, Vulpetti A, Ciomei M. Brasca MG, et al. Among authors: quartieri f. J Med Chem. 2009 Aug 27;52(16):5152-63. doi: 10.1021/jm9006559. J Med Chem. 2009. PMID: 19603809
A straightforward total synthesis of (-)-chaetominine.
Malgesini B, Forte B, Borghi D, Quartieri F, Gennari C, Papeo G. Malgesini B, et al. Among authors: quartieri f. Chemistry. 2009 Aug 10;15(32):7922-7929. doi: 10.1002/chem.200900793. Chemistry. 2009. PMID: 19562787