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Page 1
Di-bromo-Based Small-Molecule Inhibitors of the PD-1/PD-L1 Immune Checkpoint.
J Med Chem. 2020 Oct 8;63(19):11271-11285. doi: 10.1021/acs.jmedchem.0c01260. Epub 2020 Sep 23.
J Med Chem. 2020.
PMID: 32936638
Free PMC article.
Bioactive Macrocyclic Inhibitors of the PD-1/PD-L1 Immune Checkpoint.
Magiera-Mularz K, Skalniak L, Zak KM, Musielak B, Rudzinska-Szostak E, Berlicki Ł, Kocik J, Grudnik P, Sala D, Zarganes-Tzitzikas T, Shaabani S, Dömling A, Dubin G, Holak TA.
Magiera-Mularz K, et al. Among authors: sala d.
Angew Chem Int Ed Engl. 2017 Oct 23;56(44):13732-13735. doi: 10.1002/anie.201707707. Epub 2017 Sep 26.
Angew Chem Int Ed Engl. 2017.
PMID: 28881104
Free PMC article.
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Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction.
Muszak D, Surmiak E, Plewka J, Magiera-Mularz K, Kocik-Krol J, Musielak B, Sala D, Kitel R, Stec M, Weglarczyk K, Siedlar M, Dömling A, Skalniak L, Holak TA.
Muszak D, et al. Among authors: sala d.
J Med Chem. 2021 Aug 12;64(15):11614-11636. doi: 10.1021/acs.jmedchem.1c00957. Epub 2021 Jul 27.
J Med Chem. 2021.
PMID: 34313116
Free PMC article.
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Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists.
Butera R, Ważyńska M, Magiera-Mularz K, Plewka J, Musielak B, Surmiak E, Sala D, Kitel R, de Bruyn M, Nijman HW, Elsinga PH, Holak TA, Dömling A.
Butera R, et al. Among authors: sala d.
ACS Med Chem Lett. 2021 Apr 28;12(5):768-773. doi: 10.1021/acsmedchemlett.1c00033. eCollection 2021 May 13.
ACS Med Chem Lett. 2021.
PMID: 34055224
Free PMC article.
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CA-170 - A Potent Small-Molecule PD-L1 Inhibitor or Not?
Musielak B, Kocik J, Skalniak L, Magiera-Mularz K, Sala D, Czub M, Stec M, Siedlar M, Holak TA, Plewka J.
Musielak B, et al. Among authors: sala d.
Molecules. 2019 Aug 1;24(15):2804. doi: 10.3390/molecules24152804.
Molecules. 2019.
PMID: 31374878
Free PMC article.
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Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions.
Musielak B, Janczyk W, Rodriguez I, Plewka J, Sala D, Magiera-Mularz K, Holak T.
Musielak B, et al. Among authors: sala d.
Molecules. 2020 Jul 1;25(13):3017. doi: 10.3390/molecules25133017.
Molecules. 2020.
PMID: 32630327
Free PMC article.
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Human and mouse PD-L1: similar molecular structure, but different druggability profiles.
Magiera-Mularz K, Kocik J, Musielak B, Plewka J, Sala D, Machula M, Grudnik P, Hajduk M, Czepiel M, Siedlar M, Holak TA, Skalniak L.
Magiera-Mularz K, et al. Among authors: sala d.
iScience. 2020 Dec 24;24(1):101960. doi: 10.1016/j.isci.2020.101960. eCollection 2021 Jan 22.
iScience. 2020.
PMID: 33437940
Free PMC article.
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