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Page 1
Structure-Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis.
Dichiara M, Simpson QJ, Quotadamo A, Jalani HB, Huang AX, Millard CC, Klug DM, Tse EG, Todd MH, Silva DG, da Silva Emery F, Carlson JE, Zheng SL, Vleminckx M, Matheeussen A, Caljon G, Pollastri MP, Sjö P, Perry B, Ferrins L. Dichiara M, et al. ACS Infect Dis. 2023 Aug 11;9(8):1470-1487. doi: 10.1021/acsinfecdis.3c00040. Epub 2023 Jul 7. ACS Infect Dis. 2023. PMID: 37417544 Free PMC article.
Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus.
Klug DM, Tse EG, Silva DG, Cao Y, Charman SA, Chauhan J, Crighton E, Dichiara M, Drake C, Drewry D, da Silva Emery F, Ferrins L, Graves L, Hopkins E, Kresina TAC, Lorente-Macías Á, Perry B, Phipps R, Quiroga B, Quotadamo A, Sabatino GN, Sama A, Schätzlein A, Simpson QJ, Steele J, Shanu-Wilson J, Sjö P, Stapleton P, Swain CJ, Vaideanu A, Xie H, Zuercher W, Todd MH. Klug DM, et al. Among authors: silva dg. ACS Infect Dis. 2023 Dec 8;9(12):2423-2435. doi: 10.1021/acsinfecdis.3c00286. Epub 2023 Nov 22. ACS Infect Dis. 2023. PMID: 37991879 Free PMC article.
New Class of Antitrypanosomal Agents Based on Imidazopyridines.
Silva DG, Gillespie JR, Ranade RM, Herbst ZM, Nguyen UTT, Buckner FS, Montanari CA, Gelb MH. Silva DG, et al. ACS Med Chem Lett. 2017 Jun 27;8(7):766-770. doi: 10.1021/acsmedchemlett.7b00202. eCollection 2017 Jul 13. ACS Med Chem Lett. 2017. PMID: 28740614 Free PMC article.
On the intrinsic reactivity of highly potent trypanocidal cruzain inhibitors.
Bonatto V, Batista PHJ, Cianni L, De Vita D, Silva DG, Cedron R, Tezuka DY, de Albuquerque S, Moraes CB, Franco CH, Lameira J, Leitão A, Montanari CA. Bonatto V, et al. Among authors: silva dg. RSC Med Chem. 2020 Sep 9;11(11):1275-1284. doi: 10.1039/d0md00097c. eCollection 2020 Nov 18. RSC Med Chem. 2020. PMID: 34095840 Free PMC article.
Development of the First Potential Nonpeptidic Positron Emission Tomography Tracer for the Imaging of CCR2 Receptors.
Wagner S, de Moura Gatti F, Silva DG, Ortiz Zacarias NV, Zweemer AJM, Hermann S, De Maria M, Koch M, Weiss C, Schepmann D, Heitman LH, Tschammer N, Kopka K, Junker A. Wagner S, et al. Among authors: silva dg. ChemMedChem. 2021 Feb 17;16(4):640-645. doi: 10.1002/cmdc.202000728. Epub 2020 Nov 23. ChemMedChem. 2021. PMID: 33205603 Free PMC article.
14 results