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2017 1
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2019 6
2020 6
2021 3
2022 6
2023 3
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26 results

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Page 1
The mechanisms of pharmacokinetic food-drug interactions - A perspective from the UNGAP group.
Koziolek M, Alcaro S, Augustijns P, Basit AW, Grimm M, Hens B, Hoad CL, Jedamzik P, Madla CM, Maliepaard M, Marciani L, Maruca A, Parrott N, Pávek P, Porter CJH, Reppas C, van Riet-Nales D, Rubbens J, Statelova M, Trevaskis NL, Valentová K, Vertzoni M, Čepo DV, Corsetti M. Koziolek M, et al. Among authors: maruca a. Eur J Pharm Sci. 2019 Jun 15;134:31-59. doi: 10.1016/j.ejps.2019.04.003. Epub 2019 Apr 8. Eur J Pharm Sci. 2019. PMID: 30974173 Free article. Review.
Mapping Chromone-3-Phenylcarboxamide Pharmacophore: Quid Est Veritas?
Mesiti F, Gaspar A, Chavarria D, Maruca A, Rocca R, Gil Martins E, Barreiro S, Silva R, Fernandes C, Gul S, Keminer O, Alcaro S, Borges F. Mesiti F, et al. Among authors: maruca a. J Med Chem. 2021 Aug 12;64(15):11169-11182. doi: 10.1021/acs.jmedchem.1c00510. Epub 2021 Jul 16. J Med Chem. 2021. PMID: 34269579
4-Oxoquinolines and monoamine oxidase: When tautomerism matters.
Mesiti F, Maruca A, Silva V, Rocca R, Fernandes C, Remião F, Uriarte E, Alcaro S, Gaspar A, Borges F. Mesiti F, et al. Among authors: maruca a. Eur J Med Chem. 2021 Mar 5;213:113183. doi: 10.1016/j.ejmech.2021.113183. Epub 2021 Jan 13. Eur J Med Chem. 2021. PMID: 33493825
Identification of SET/EED dual binders as innovative PRC2 inhibitors.
Catalano R, Maruca A, Rocca R, Tassone P, Panzarella G, Costa G, Ortuso F, Alcaro S. Catalano R, et al. Among authors: maruca a. Future Med Chem. 2022 May;14(9):609-621. doi: 10.4155/fmc-2022-0010. Epub 2022 Mar 29. Future Med Chem. 2022. PMID: 35348013
Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis.
Albertini C, Salerno A, Atzeni S, Uliassi E, Massenzio F, Maruca A, Rocca R, Mecava M, Silva FSG, Mena D, Valente P, Duarte AI, Chavarria D, Bissaro M, Moro S, Federico S, Spalluto G, Soukup O, Borges F, Alcaro S, Monti B, Oliveira PJ, Menéndez JC, Bolognesi ML. Albertini C, et al. Among authors: maruca a. ACS Chem Neurosci. 2022 Aug 3;13(15):2252-2260. doi: 10.1021/acschemneuro.2c00261. Epub 2022 Jul 22. ACS Chem Neurosci. 2022. PMID: 35868251 Free PMC article.
Discovery of first novel sigma/HDACi dual-ligands with a potent in vitro antiproliferative activity.
Barbaraci C, di Giacomo V, Maruca A, Patamia V, Rocca R, Dichiara M, Di Rienzo A, Cacciatore I, Cataldi A, Balaha M, Rapino M, Zagni C, Zampieri D, Pasquinucci L, Parenti C, Amata E, Rescifina A, Alcaro S, Marrazzo A. Barbaraci C, et al. Among authors: maruca a. Bioorg Chem. 2023 Nov;140:106794. doi: 10.1016/j.bioorg.2023.106794. Epub 2023 Aug 23. Bioorg Chem. 2023. PMID: 37659146 Free article.
26 results