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Page 1
Synthesis of cinnamic acid derivatives and leishmanicidal activity against Leishmania braziliensis.
Rodrigues MP, Tomaz DC, Ângelo de Souza L, Onofre TS, Aquiles de Menezes W, Almeida-Silva J, Suarez-Fontes AM, Rogéria de Almeida M, Manoel da Silva A, Bressan GC, Vannier-Santos MA, Rangel Fietto JL, Teixeira RR. Rodrigues MP, et al. Among authors: teixeira rr. Eur J Med Chem. 2019 Dec 1;183:111688. doi: 10.1016/j.ejmech.2019.111688. Epub 2019 Sep 9. Eur J Med Chem. 2019. PMID: 31542714
Synthesis of vanillin derivatives with 1,2,3-triazole fragments and evaluation of their fungicide and fungistatic activities.
Gazolla PAR, de Aguiar AR, Costa MCA, Oliveira OV, Costa AV, da Silva CM, do Nascimento CJ, Junker J, Ferreira RS, de Oliveira FM, Vaz BG, do Carmo PHF, Santos DA, Ferreira MMC, Teixeira RR. Gazolla PAR, et al. Among authors: teixeira rr. Arch Pharm (Weinheim). 2023 Jun;356(6):e2200653. doi: 10.1002/ardp.202200653. Epub 2023 Mar 15. Arch Pharm (Weinheim). 2023. PMID: 36922908
Novel diamides inspired by protein kinase inhibitors as anti-Trypanosoma cruzi agents: in vitro and in vivo evaluations.
Vieira da Silva Torchelsen FK, Fernandes Pedrosa TC, Rodrigues MP, de Aguiar AR, de Oliveira FM, Amarante GW, Sales-Junior PA, Branquinho RT, Gomes da Silva SP, Talvani A, Fonseca Murta SM, Martins FT, Braun RL, Teixeira RR, Furtado Mosqueira VC, Lana M. Vieira da Silva Torchelsen FK, et al. Among authors: teixeira rr. Future Med Chem. 2023 Aug;15(16):1469-1489. doi: 10.4155/fmc-2023-0090. Epub 2023 Aug 31. Future Med Chem. 2023. PMID: 37650735
In vitro evaluation of antileishmanial activity, mode of action and cellular response induced by vanillin synthetic derivatives against Leishmania species able to cause cutaneous and visceral leishmaniasis.
Freitas CS, Santiago SS, Lage DP, Antinarelli LMR, Oliveira FM, Vale DL, Martins VT, Magalhaes LND, Bandeira RS, Ramos FF, Pereira IAG, de Jesus MM, Ludolf F, Tavares GSV, Costa AV, Ferreira RS, Coimbra ES, Teixeira RR, Coelho EAF. Freitas CS, et al. Among authors: teixeira rr. Exp Parasitol. 2023 Aug;251:108555. doi: 10.1016/j.exppara.2023.108555. Epub 2023 May 27. Exp Parasitol. 2023. PMID: 37247802
The SRPK inhibitor N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl) isonicotinamide (SRPIN340) increases the immune response against metastatic melanoma in mice.
Moreira GA, Caetano MMM, do Vale JA, de Paiva JC, Gonçalves VHS, Almeida AA, Silva LVG, Martim FRG, de Andrade Barros MV, Guimarães GR, de Oliveira Santos L, de Souza APM, Machado-Neves M, Teixeira RR, Silva-Júnior A, Fietto JLR, Boroni M, de Oliveira LL, Bressan GC. Moreira GA, et al. Among authors: teixeira rr. Biochem Pharmacol. 2022 Sep;203:115161. doi: 10.1016/j.bcp.2022.115161. Epub 2022 Jul 2. Biochem Pharmacol. 2022. PMID: 35787994 Free article.
Antimetastatic effect of the pharmacological inhibition of serine/arginine-rich protein kinases (SRPK) in murine melanoma.
Moreira GA, Lima GDA, Siqueira RP, Barros MVA, Adjanohoun ALM, Santos VC, Barbosa ÉAA, Loterio RK, Paiva JC, Gonçalves VHS, Viol LCS, Marques-da-Silva EA, Júnior AS, Almeida MR, Fietto JLR, Machado-Neves M, Ferreira RS, Teixeira RR, Bressan GC. Moreira GA, et al. Among authors: teixeira rr. Toxicol Appl Pharmacol. 2018 Oct 1;356:214-223. doi: 10.1016/j.taap.2018.08.012. Epub 2018 Aug 20. Toxicol Appl Pharmacol. 2018. PMID: 30138656 Free article.
Immunomodulatory activity of trifluoromethyl arylamides derived from the SRPK inhibitor SRPIN340 and their potential use as vaccine adjuvant.
Mendes FC, de Paiva JC, da Silva EQG, Santos MR, de Almeida Lima GD, Moreira GA, Silva LVG, de Melo Agripino J, de Souza APM, de Oliveira Mendes TA, Machado-Neves M, Teixeira RR, Silva-Júnior A, Fietto JLR, de Oliveira LL, Bressan GC. Mendes FC, et al. Among authors: teixeira rr. Life Sci. 2022 Oct 15;307:120849. doi: 10.1016/j.lfs.2022.120849. Epub 2022 Aug 1. Life Sci. 2022. PMID: 35926588 Free article.
In vitro tripanocidal effect of 1,8-dioxooctahydroxanthenes (xanthenodiones) and tetraketones and improvement of cardiac parameters in vivo.
Menezes APJ, Silva MLD, Pereira WL, Costa GP, Horta AL, Mendonça AAS, Carneiro ACA, Souza DMS, Novaes RD, Teixeira RR, Talvani A. Menezes APJ, et al. Among authors: teixeira rr. J Glob Antimicrob Resist. 2020 Sep;22:466-476. doi: 10.1016/j.jgar.2020.04.005. Epub 2020 May 14. J Glob Antimicrob Resist. 2020. PMID: 32417591 Free article.
105 results