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Amide-to-Triazole Switch in Somatostatin-14-Based Radioligands: Impact on Receptor Affinity and In Vivo Stability.
Pharmaceutics. 2024 Mar 13;16(3):392. doi: 10.3390/pharmaceutics16030392.
Pharmaceutics. 2024.
PMID: 38543286
Free PMC article.
Straightforward Synthesis of DFO* - An Octadentate Chelator for Zirconium-89.
Guarrochena X, Kronberger J, Tieber M, Ciesielski P, Mindt TL, Feiner IVJ.
Guarrochena X, et al.
ChemMedChem. 2024 Feb 1;19(3):e202300495. doi: 10.1002/cmdc.202300495. Epub 2024 Jan 11.
ChemMedChem. 2024.
PMID: 38102942
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Automated solid-phase synthesis of metabolically stabilized triazolo-peptidomimetics.
Guarrochena X, Kaudela B, Mindt TL.
Guarrochena X, et al.
J Pept Sci. 2023 Sep;29(9):e3488. doi: 10.1002/psc.3488. Epub 2023 Mar 29.
J Pept Sci. 2023.
PMID: 36912359
Free PMC article.
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Mini-review: Targeted radiopharmaceuticals incorporating reversible, low molecular weight albumin binders.
Brandt M, Cardinale J, Giammei C, Guarrochena X, Happl B, Jouini N, Mindt TL.
Brandt M, et al. Among authors: guarrochena x.
Nucl Med Biol. 2019 Mar;70:46-52. doi: 10.1016/j.nucmedbio.2019.01.006. Epub 2019 Jan 26.
Nucl Med Biol. 2019.
PMID: 30831342
Review.
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