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Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase-2 (SHP2).
J Med Chem. 2024 Mar 28;67(6):4655-4675. doi: 10.1021/acs.jmedchem.3c02118. Epub 2024 Mar 10.
J Med Chem. 2024.
PMID: 38462716
Fragment-to-Lead Medicinal Chemistry Publications in 2022.
Woodhead AJ, Erlanson DA, de Esch IJP, Holvey RS, Jahnke W, Pathuri P.
Woodhead AJ, et al. Among authors: holvey rs.
J Med Chem. 2024 Feb 22;67(4):2287-2304. doi: 10.1021/acs.jmedchem.3c02070. Epub 2024 Jan 30.
J Med Chem. 2024.
PMID: 38289623
Review.
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C-H functionalisation tolerant to polar groups could transform fragment-based drug discovery (FBDD).
Chessari G, Grainger R, Holvey RS, Ludlow RF, Mortenson PN, Rees DC.
Chessari G, et al. Among authors: holvey rs.
Chem Sci. 2021 Sep 1;12(36):11976-11985. doi: 10.1039/d1sc03563k. eCollection 2021 Sep 22.
Chem Sci. 2021.
PMID: 34667563
Free PMC article.
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Structure-Based Design of Potent and Orally Active Isoindolinone Inhibitors of MDM2-p53 Protein-Protein Interaction.
Chessari G, Hardcastle IR, Ahn JS, Anil B, Anscombe E, Bawn RH, Bevan LD, Blackburn TJ, Buck I, Cano C, Carbain B, Castro J, Cons B, Cully SJ, Endicott JA, Fazal L, Golding BT, Griffin RJ, Haggerty K, Harnor SJ, Hearn K, Hobson S, Holvey RS, Howard S, Jennings CE, Johnson CN, Lunec J, Miller DC, Newell DR, Noble MEM, Reeks J, Revill CH, Riedinger C, St Denis JD, Tamanini E, Thomas H, Thompson NT, Vinković M, Wedge SR, Williams PA, Wilsher NE, Zhang B, Zhao Y.
Chessari G, et al. Among authors: holvey rs.
J Med Chem. 2021 Apr 8;64(7):4071-4088. doi: 10.1021/acs.jmedchem.0c02188. Epub 2021 Mar 24.
J Med Chem. 2021.
PMID: 33761253
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Selective Targeting of the TPX2 Site of Importin-α Using Fragment-Based Ligand Design.
Holvey RS, Valkov E, Neal D, Stewart M, Abell C.
Holvey RS, et al.
ChemMedChem. 2015 Jul;10(7):1232-9. doi: 10.1002/cmdc.201500014. Epub 2015 Apr 20.
ChemMedChem. 2015.
PMID: 25899172
Free PMC article.
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