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Exploring Hydrophilic PD-L1 Radiotracers Utilizing Phosphonic Acids: Insights into Unforeseen Pharmacokinetics.
Int J Mol Sci. 2023 Oct 11;24(20):15088. doi: 10.3390/ijms242015088.
Int J Mol Sci. 2023.
PMID: 37894769
Free PMC article.
Development of Radiotracers for Imaging of the PD-1/PD-L1 Axis.
Krutzek F, Kopka K, Stadlbauer S.
Krutzek F, et al.
Pharmaceuticals (Basel). 2022 Jun 14;15(6):747. doi: 10.3390/ph15060747.
Pharmaceuticals (Basel). 2022.
PMID: 35745666
Free PMC article.
Review.
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Design and Biological Evaluation of Small-Molecule PET-Tracers for Imaging of Programmed Death Ligand 1.
Krutzek F, Donat CK, Ullrich M, Zarschler K, Ludik MC, Feldmann A, Loureiro LR, Kopka K, Stadlbauer S.
Krutzek F, et al.
Cancers (Basel). 2023 May 6;15(9):2638. doi: 10.3390/cancers15092638.
Cancers (Basel). 2023.
PMID: 37174103
Free PMC article.
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Design, Synthesis, and Biological Evaluation of Small-Molecule-Based Radioligands with Improved Pharmacokinetic Properties for Imaging of Programmed Death Ligand 1.
Krutzek F, Donat CK, Ullrich M, Stadlbauer S.
Krutzek F, et al.
J Med Chem. 2023 Dec 14;66(23):15894-15915. doi: 10.1021/acs.jmedchem.3c01355. Epub 2023 Dec 1.
J Med Chem. 2023.
PMID: 38038981
Free PMC article.
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Chelator impact: investigating the pharmacokinetic behavior of copper-64 labeled PD-L1 radioligands.
Krutzek F, Donat CK, Stadlbauer S.
Krutzek F, et al.
EJNMMI Radiopharm Chem. 2024 Feb 19;9(1):14. doi: 10.1186/s41181-024-00243-5.
EJNMMI Radiopharm Chem. 2024.
PMID: 38372838
Free PMC article.
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K-Region-Extended [c]-Heteroannulated Pyrenes.
Baumgärtner K, Kirschbaum T, Krutzek F, Dreuw A, Rominger F, Mastalerz M.
Baumgärtner K, et al. Among authors: krutzek f.
Chemistry. 2017 Dec 14;23(70):17817-17822. doi: 10.1002/chem.201703988. Epub 2017 Nov 16.
Chemistry. 2017.
PMID: 28977702
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