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Page 1
Effect of metformin in hypothalamic astrocytes from an immunocompromised mice model.
Bobermin LD, da Costa DS, de Moraes ADM, da Silva VF, de Oliveira GT, Sesterheim P, Tramontina AC, Basso LA, Leipnitz G, Quincozes-Santos A, Gonçalves CA. Bobermin LD, et al. Among authors: basso la. Biochimie. 2024 Apr 18:S0300-9084(24)00080-4. doi: 10.1016/j.biochi.2024.04.005. Online ahead of print. Biochimie. 2024. PMID: 38642825
Exploring Scaffold Hopping for Novel 2-(Quinolin-4-yloxy)acetamides with Enhanced Antimycobacterial Activity.
Borsoi AF, Silva Ramos A, Sperotto N, Abbadi BL, Souza Macchi Hopf F, da Silva Dadda A, Scheibler Rambo R, Neves Muniz M, Delgado Paz J, Silveira Grams E, Fries da Silva F, Pissinate K, Galina L, Calle González L, Silva Duarte L, Alberton Perelló M, de Matos Czeczot A, Bizarro CV, Basso LA, Machado P. Borsoi AF, et al. Among authors: basso la. ACS Med Chem Lett. 2024 Mar 11;15(4):493-500. doi: 10.1021/acsmedchemlett.3c00570. eCollection 2024 Apr 11. ACS Med Chem Lett. 2024. PMID: 38628799
SARS-CoV-2 immune complex triggers human monocyte necroptosis.
Santos LD, Antunes KH, Cassão G, Gonçalves JI, Abbadi BL, Bizarro CV, Basso LA, Machado P, de Souza APD, Porto BN. Santos LD, et al. Among authors: basso la. Int Immunopharmacol. 2023 Apr;117:109954. doi: 10.1016/j.intimp.2023.109954. Epub 2023 Feb 27. Int Immunopharmacol. 2023. PMID: 36870284 Free PMC article.
Identification of potential inhibitors of Mycobacterium tuberculosis shikimate kinase: molecular docking, in silico toxicity and in vitro experiments.
Freitas de Freitas T, Roth CD, Abbadi BL, Hopf FSM, Perelló MA, de Matos Czeczot A, de Souza EV, Borsoi AF, Machado P, Bizarro CV, Basso LA, Timmers LFSM. Freitas de Freitas T, et al. Among authors: basso la. J Comput Aided Mol Des. 2023 Mar;37(3):117-128. doi: 10.1007/s10822-022-00495-w. Epub 2022 Dec 22. J Comput Aided Mol Des. 2023. PMID: 36547753 Free PMC article.
Novel 4-aminoquinolines: Synthesis, inhibition of the Mycobacterium tuberculosis enoyl-acyl carrier protein reductase, antitubercular activity, SAR, and preclinical evaluation.
Paz JD, Denise de Moura Sperotto N, Ramos AS, Pissinate K, da Silva Rodrigues Junior V, Abbadi BL, Borsoi AF, Rambo RS, Corso Minotto AC, da Silva Dadda A, Galina L, Macchi Hopf FS, Muniz MN, Borges Martinelli LK, Roth CD, Madeira Silva RB, Perelló MA, de Matos Czeczot A, Neves CE, Duarte LS, Leyser M, Dias de Oliveira S, Bizarro CV, Machado P, Basso LA. Paz JD, et al. Among authors: basso la. Eur J Med Chem. 2023 Jan 5;245(Pt 1):114908. doi: 10.1016/j.ejmech.2022.114908. Epub 2022 Nov 18. Eur J Med Chem. 2023. PMID: 36435016
Antitubercular Activity of Novel 2-(Quinoline-4-yloxy)acetamides with Improved Drug-Like Properties.
Borsoi AF, Alice LM, Sperotto N, Ramos AS, Abbadi BL, Macchi Hopf FS, Silva Dadda AD, Rambo RS, Madeira Silva RB, Paz JD, Pissinate K, Muniz MN, Neves CE, Galina L, González LC, Perelló MA, de Matos Czeczot A, Leyser M, de Oliveira SD, de Araújo Lock G, de Araújo BV, Costa TD, Bizarro CV, Basso LA, Machado P. Borsoi AF, et al. Among authors: basso la. ACS Med Chem Lett. 2022 Jul 21;13(8):1337-1344. doi: 10.1021/acsmedchemlett.2c00254. eCollection 2022 Aug 11. ACS Med Chem Lett. 2022. PMID: 35978694 Free PMC article.
Evaluation of 3-Deoxy-D-Arabino-Heptulosonate 7-Phosphate Synthase (DAHPS) as a Vulnerable Target in Mycobacterium tuberculosis.
Galina L, Hopf FSM, Abbadi BL, Sperotto NDM, Czeczot AM, Duque-Villegas MA, Perello MA, Matter LB, de Souza EV, Parish T, Machado P, Basso LA, Bizarro CV. Galina L, et al. Among authors: basso la. Microbiol Spectr. 2022 Aug 31;10(4):e0072822. doi: 10.1128/spectrum.00728-22. Epub 2022 Jul 14. Microbiol Spectr. 2022. PMID: 35862980 Free PMC article.
191 results