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Potentiating-antibiotic activity and absorption, distribution, metabolism, excretion and toxicity properties (ADMET) analysis of synthetic thiadiazines against multi-drug resistant (MDR) strains.
de Araújo ACJ, Freitas PR, Araújo IM, Siqueira GM, de Oliveira Borges JA, Alves DS, Miranda GM, Dos Santos Nascimento IJ, de Araújo-Júnior JX, da Silva-Júnior EF, de Aquino TM, Junior FJBM, Marinho ES, Dos Santos HS, Tintino SR, Coutinho HDM. de Araújo ACJ, et al. Among authors: de aquino tm. Fundam Clin Pharmacol. 2024 Feb;38(1):84-98. doi: 10.1111/fcp.12950. Epub 2023 Aug 30. Fundam Clin Pharmacol. 2024. PMID: 37649138
Synthesis, anti-Toxoplasma gondii and antimicrobial activities of benzaldehyde 4-phenyl-3-thiosemicarbazones and 2-[(phenylmethylene)hydrazono]-4-oxo-3-phenyl-5-thiazolidineacetic acids.
de Aquino TM, Liesen AP, da Silva RE, Lima VT, Carvalho CS, de Faria AR, de Araújo JM, de Lima JG, Alves AJ, de Melo EJ, Góes AJ. de Aquino TM, et al. Among authors: de melo ej, de araujo jm, de lima jg, de faria ar. Bioorg Med Chem. 2008 Jan 1;16(1):446-56. doi: 10.1016/j.bmc.2007.09.025. Epub 2007 Sep 18. Bioorg Med Chem. 2008. PMID: 17905587
Dynamic Simulation, Docking and DFT Studies Applied to a Set of Anti-Acetylcholinesterase Inhibitors in the enzyme β-Secretase (BACE-1): An Important Therapeutic Target in Alzheimer`s disease.
Silva-Junior EF, Barcellos Franca PH, Quintans-Junior LJ, Mendonca-Junior FJB, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. Silva-Junior EF, et al. Among authors: de araujo junior jx, de aquino tm. Curr Comput Aided Drug Des. 2017 Nov 10;13(4):266-274. doi: 10.2174/1573409913666170406150905. Curr Comput Aided Drug Des. 2017. PMID: 28382866
Molecular Docking Studies Applied to a Dataset of Cruzain Inhibitors.
da Silva-Junior EF, Barcellos Franca PH, Ribeiro FF, Bezerra Mendonca-Junior FJ, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. da Silva-Junior EF, et al. Among authors: de araujo junior jx, de aquino tm. Curr Comput Aided Drug Des. 2018;14(1):68-78. doi: 10.2174/1573409913666170519112758. Curr Comput Aided Drug Des. 2018. PMID: 28523999
Aminoguanidine hydrazones (AGH's) as modulators of norfloxacin resistance in Staphylococcus aureus that overexpress NorA efflux pump.
Dantas N, de Aquino TM, de Araújo-Júnior JX, da Silva-Júnior E, Gomes EA, Gomes AAS, Siqueira-Júnior JP, Mendonça Junior FJB. Dantas N, et al. Among authors: de araujo junior jx, de aquino tm. Chem Biol Interact. 2018 Jan 25;280:8-14. doi: 10.1016/j.cbi.2017.12.009. Epub 2017 Dec 5. Chem Biol Interact. 2018. PMID: 29208359
Annonalide and derivatives: Semisynthesis, cytotoxic activities and studies on interaction of annonalide with DNA.
Marques RA, Gomes AOCV, de Brito MV, Dos Santos ALP, da Silva GS, de Lima LB, Nunes FM, de Mattos MC, de Oliveira FCE, do Ó Pessoa C, de Moraes MO, de Fátima Â, Franco LL, Silva MM, Dantas MDA, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, de Oliveira MCF, Leslie Gunatilaka AA. Marques RA, et al. Among authors: de araujo junior jx, de aquino tm, de oliveira mcf, de lima lb, de mattos mc, de moraes mo, de fatima a, de oliveira fce, de brito mv. J Photochem Photobiol B. 2018 Feb;179:156-166. doi: 10.1016/j.jphotobiol.2018.01.016. Epub 2018 Feb 3. J Photochem Photobiol B. 2018. PMID: 29413989
Evidence for the involvement of TNF-α, IL-1β and IL-10 in the antinociceptive and anti-inflammatory effects of indole-3-guanylhydrazone hydrochloride, an aromatic aminoguanidine, in rodents.
Sandes SMS, Heimfarth L, Brito RG, Santos PL, Gouveia DN, Carvalho AMS, Quintans JSS, da Silva-Júnior EF, de Aquino TM, França PHB, de Araújo-Júnior JX, Albuquerque-Júnior RLC, Zengin G, Schmitt M, Bourguignon JJ, Quintans-Júnior LJ. Sandes SMS, et al. Among authors: de araujo junior jx, de aquino tm. Chem Biol Interact. 2018 Apr 25;286:1-10. doi: 10.1016/j.cbi.2018.02.026. Epub 2018 Feb 27. Chem Biol Interact. 2018. PMID: 29499192
Highly functionalized piperidines: Free radical scavenging, anticancer activity, DNA interaction and correlation with biological activity.
Das S, da Silva CJ, Silva MM, Dantas MDA, de Fátima Â, Góis Ruiz ALT, da Silva CM, de Carvalho JE, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, Brahmachari G, Modolo LV. Das S, et al. Among authors: de araujo junior jx, de aquino tm, de fatima a, de carvalho je. J Adv Res. 2017 Oct 31;9:51-61. doi: 10.1016/j.jare.2017.10.010. eCollection 2018 Jan. J Adv Res. 2017. PMID: 30046486 Free PMC article.
Correlation between DNA/HSA-interactions and antimalarial activity of acridine derivatives: Proposing a possible mechanism of action.
de M Silva M, Macedo TS, Teixeira HMP, Moreira DRM, Soares MBP, da C Pereira AL, de L Serafim V, Mendonça-Júnior FJB, do Carmo A de Lima M, de Moura RO, da Silva-Júnior EF, de Araújo-Júnior JX, de A Dantas MD, de O O Nascimento E, Maciel TMS, de Aquino TM, Figueiredo IM, Santos JCC. de M Silva M, et al. Among authors: de araujo junior jx, de o o nascimento e, de moura ro, de aquino tm, de a dantas md, de l serafim v. J Photochem Photobiol B. 2018 Dec;189:165-175. doi: 10.1016/j.jphotobiol.2018.10.016. Epub 2018 Oct 19. J Photochem Photobiol B. 2018. PMID: 30366283
5-Nitro-Thiophene-Thiosemicarbazone Derivatives Present Antitumor Activity Mediated by Apoptosis and DNA Intercalation.
Roque Marques KM, do Desterro MR, de Arruda SM, de Araújo Neto LN, do Carmo Alves de Lima M, de Almeida SMV, da Silva ECD, de Aquino TM, da Silva-Júnior EF, de Araújo-Júnior JX, de M Silva M, de A Dantas MD, Santos JCC, Figueiredo IM, Bazin MA, Marchand P, da Silva TG, Mendonça Junior FJB. Roque Marques KM, et al. Among authors: de almeida smv, de araujo junior jx, de aquino tm, de a dantas md, de m silva m, de arruda sm, de araujo neto ln. Curr Top Med Chem. 2019;19(13):1075-1091. doi: 10.2174/1568026619666190621120304. Curr Top Med Chem. 2019. PMID: 31223089
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