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Novel VEGFR2 inhibitors with thiazoloquinoxaline scaffold targeting hepatocellular carcinoma with lower cardiotoxic impact.
Sci Rep. 2023 Aug 25;13(1):13907. doi: 10.1038/s41598-023-40832-z.
Sci Rep. 2023.
PMID: 37626064
Free PMC article.
Novel thioureido-benzenesulfonamide derivatives with enaminone linker as potent anticancer, radiosensitizers and VEGFR2 inhibitors.
Ghorab MM, Ragab FA, Heiba HI, El-Gazzar MG, El-Gazzar MGM.
Ghorab MM, et al. Among authors: el gazzar mgm.
Bioorg Med Chem Lett. 2018 May 15;28(9):1464-1470. doi: 10.1016/j.bmcl.2018.03.089. Epub 2018 Mar 31.
Bioorg Med Chem Lett. 2018.
PMID: 29628325
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Computational, in vitro and radiation-based in vivo studies on acetamide quinazolinone derivatives as new proposed purine nucleoside phosphorylase inhibitors for breast cancer.
El-Gazzar MGM, Ghorab MM, Amin MA, Korany M, Khedr MA, El-Gazzar MG, Sakr TM.
El-Gazzar MGM, et al.
Eur J Med Chem. 2023 Feb 15;248:115087. doi: 10.1016/j.ejmech.2023.115087. Epub 2023 Jan 2.
Eur J Med Chem. 2023.
PMID: 36610250
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Quinazolinone derivatives as new potential CDK4/6 inhibitors, apoptosis inducers and radiosensitizers for breast cancer.
El-Gazzar MG, El-Gazzar MG, Ghorab MM.
El-Gazzar MG, et al.
Future Med Chem. 2023 Jul;15(13):1133-1147. doi: 10.4155/fmc-2023-0126. Epub 2023 Aug 2.
Future Med Chem. 2023.
PMID: 37529897
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Synthesis, in-vitro anticancer screening and radiosensitizing evaluation of some new N-(quinoxalin-2-yl)benzenesulfonamide derivatives.
Ghorab MM, Ragab FA, Heiba HI, El-Gazzar MG, El-Gazzar MG.
Ghorab MM, et al.
Arzneimittelforschung. 2012 Jan;62(1):46-52. doi: 10.1055/s-0031-1295496. Epub 2012 Jan 10.
Arzneimittelforschung. 2012.
PMID: 22331763
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