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Structure activity relationships of 5-HT2B and 5-HT2C serotonin receptor antagonists: N6, C2 and 5'-Modified (N)-methanocarba-adenosine derivatives.
Eur J Med Chem. 2023 Nov 5;259:115691. doi: 10.1016/j.ejmech.2023.115691. Epub 2023 Jul 31.
Eur J Med Chem. 2023.
PMID: 37562117
Synthesis and pharmacological characterization of multiply substituted 2H-chromene derivatives as P2Y6 receptor antagonists.
Jung YH, Shah Q, Lewicki SA, Pramanik A, Gopinatth V, Pelletier J, Sévigny J, Iqbal J, Jacobson KA.
Jung YH, et al. Among authors: lewicki sa.
Bioorg Med Chem Lett. 2022 Nov 1;75:128981. doi: 10.1016/j.bmcl.2022.128981. Epub 2022 Sep 8.
Bioorg Med Chem Lett. 2022.
PMID: 36089113
Free PMC article.
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Structure-Activity Relationship and Neuroprotective Activity of 1,5-Dihydro-2H-naphtho[1,2-b][1,4]diazepine-2,4(3H)-diones as P2X4 Receptor Antagonists.
Toti KS, Verma R, McGonnigle MJ, Gamiotea Turro D, Wen Z, Lewicki SA, Liang BT, Jacobson KA.
Toti KS, et al. Among authors: lewicki sa.
J Med Chem. 2022 Oct 27;65(20):13967-13987. doi: 10.1021/acs.jmedchem.2c01197. Epub 2022 Sep 23.
J Med Chem. 2022.
PMID: 36150180
Free PMC article.
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In vivo phenotypic validation of adenosine receptor-dependent activity of non-adenosine drugs.
Xiao C, Gavrilova O, Liu N, Lewicki SA, Reitman ML, Jacobson KA.
Xiao C, et al. Among authors: lewicki sa.
Purinergic Signal. 2023 Sep;19(3):551-564. doi: 10.1007/s11302-023-09924-3. Epub 2023 Feb 13.
Purinergic Signal. 2023.
PMID: 36781825
Free PMC article.
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Alicyclic Ring Size Variation of 4-Phenyl-2-naphthoic Acid Derivatives as P2Y14 Receptor Antagonists.
Wen Z, Pramanik A, Lewicki SA, Jung YH, Gao ZG, Randle JCR, Cronin C, Chen Z, Giancotti LA, Whitehead GS, Liang BT, Breton S, Salvemini D, Cook DN, Jacobson KA.
Wen Z, et al. Among authors: lewicki sa.
J Med Chem. 2023 Jul 13;66(13):9076-9094. doi: 10.1021/acs.jmedchem.3c00664. Epub 2023 Jun 29.
J Med Chem. 2023.
PMID: 37382926
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Stereocontrolled access to thioisosteres of nucleoside di- and triphosphates.
Zhang HJ, Ociepa M, Nassir M, Zheng B, Lewicki SA, Salmaso V, Baburi H, Nagel J, Mirza S, Bueschbell B, Al-Hroub H, Perzanowska O, Lin Z, Schmidt MA, Eastgate MD, Jacobson KA, Müller CE, Kowalska J, Jemielity J, Baran PS.
Zhang HJ, et al. Among authors: lewicki sa.
Nat Chem. 2024 Feb;16(2):249-258. doi: 10.1038/s41557-023-01347-2. Epub 2023 Oct 19.
Nat Chem. 2024.
PMID: 37857844
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Machine learning-aided search for ligands of P2Y6 and other P2Y receptors.
Puhl AC, Lewicki SA, Gao ZG, Pramanik A, Makarov V, Ekins S, Jacobson KA.
Puhl AC, et al. Among authors: lewicki sa.
Purinergic Signal. 2024 Mar 25. doi: 10.1007/s11302-024-10003-4. Online ahead of print.
Purinergic Signal. 2024.
PMID: 38526670
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