Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
7 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Aldo-Keto Reductase 1C3 Inhibitor Prodrug Improves Pharmacokinetic Profile and Demonstrates In Vivo Efficacy in a Prostate Cancer Xenograft Model.
J Med Chem. 2023 Jul 27;66(14):9894-9915. doi: 10.1021/acs.jmedchem.3c00732. Epub 2023 Jul 10.
J Med Chem. 2023.
PMID: 37428858
Functionalized Allopurinols Targeting Amyloid-Binding Alcohol Dehydrogenase Rescue Aβ-Induced Mitochondrial Dysfunction.
Morsy A, Maddeboina K, Gao J, Wang H, Valdez J, Dow LF, Wang X, Trippier PC.
Morsy A, et al. Among authors: maddeboina k.
ACS Chem Neurosci. 2022 Jul 20;13(14):2176-2190. doi: 10.1021/acschemneuro.2c00246. Epub 2022 Jul 8.
ACS Chem Neurosci. 2022.
PMID: 35802826
Item in Clipboard
LC-MS/MS method for the quantitation of a dual PI3K/BRD4 inhibitor SF2523 in mouse plasma: Application to plasma protein binding and metabolism studies.
Bala V, Chhonker YS, Morales GA, Maddeboina K, Pal D, Durden DL, Murry DJ.
Bala V, et al. Among authors: maddeboina k.
Biomed Chromatogr. 2023 Aug;37(8):e5643. doi: 10.1002/bmc.5643. Epub 2023 Apr 27.
Biomed Chromatogr. 2023.
PMID: 37042063
Item in Clipboard
Pivotal role of nitrogen heterocycles in Alzheimer's disease drug discovery.
Kumari S, Maddeboina K, Bachu RD, Boddu SHS, Trippier PC, Tiwari AK.
Kumari S, et al. Among authors: maddeboina k.
Drug Discov Today. 2022 Oct;27(10):103322. doi: 10.1016/j.drudis.2022.07.007. Epub 2022 Jul 19.
Drug Discov Today. 2022.
PMID: 35868626
Review.
Item in Clipboard
Facile Protocol for the Synthesis of Self-assembling Polyamine-based Peptide Amphiphiles (PPAs) and Related Biomaterials.
Samad MB, Maddeboina K, Rodrigues de Almeida N, Conda-Sheridan M.
Samad MB, et al. Among authors: maddeboina k.
J Vis Exp. 2018 Jun 25;(136):57908. doi: 10.3791/57908.
J Vis Exp. 2018.
PMID: 29985361
Free PMC article.
Item in Clipboard
Discovery of an Aldo-Keto reductase 1C3 (AKR1C3) degrader.
Carmona AV, Jonnalagadda S, Case AM, Maddeboina K, Jonnalagadda SK, Dow LF, Duan L, Penning TM, Trippier PC.
Carmona AV, et al. Among authors: maddeboina k.
Commun Chem. 2024 Apr 29;7(1):95. doi: 10.1038/s42004-024-01177-4.
Commun Chem. 2024.
PMID: 38684887
Free PMC article.
Item in Clipboard
Recent advances in multitarget-directed ligands via in silico drug discovery.
Maddeboina K, Yada B, Kumari S, McHale C, Pal D, Durden DL.
Maddeboina K, et al.
Drug Discov Today. 2024 Mar;29(3):103904. doi: 10.1016/j.drudis.2024.103904. Epub 2024 Jan 26.
Drug Discov Today. 2024.
PMID: 38280625
Review.
Item in Clipboard
Cite
Cite