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Development of Novel 111In/225Ac-Labeled Agent Targeting PSMA for Highly Efficient Cancer Radiotheranostics.
J Med Chem. 2023 Jun 22;66(12):8043-8053. doi: 10.1021/acs.jmedchem.3c00346. Epub 2023 Jun 7.
J Med Chem. 2023.
PMID: 37285471
Synthesis and Evaluation of Novel 111In-Labeled Picolinic Acid-Based Radioligands Containing an Albumin Binder for Development of a Radiotheranostic Platform.
Iikuni S, Tarumizu Y, Tsuchihashi S, Ohara T, Watanabe H, Ono M.
Iikuni S, et al. Among authors: tarumizu y.
Mol Pharm. 2022 Aug 1;19(8):2725-2736. doi: 10.1021/acs.molpharmaceut.2c00071. Epub 2022 Jun 25.
Mol Pharm. 2022.
PMID: 35758049
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Radiotheranostics Using a Novel 225Ac-Labeled Radioligand with Improved Pharmacokinetics Targeting Prostate-Specific Membrane Antigen.
Iikuni S, Tarumizu Y, Nakashima K, Higaki Y, Ichikawa H, Watanabe H, Ono M.
Iikuni S, et al. Among authors: tarumizu y.
J Med Chem. 2021 Sep 23;64(18):13429-13438. doi: 10.1021/acs.jmedchem.1c00772. Epub 2021 Sep 3.
J Med Chem. 2021.
PMID: 34477385
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Characterization and Optimization of Benzimidazopyrimidine and Pyridoimidazopyridine Derivatives as Tau-SPECT Probes.
Watanabe H, Kishimoto T, Kaide S, Tarumizu Y, Tatsumi H, Iikuni S, Ono M.
Watanabe H, et al. Among authors: tarumizu y.
ACS Med Chem Lett. 2021 Apr 26;12(5):805-811. doi: 10.1021/acsmedchemlett.1c00071. eCollection 2021 May 13.
ACS Med Chem Lett. 2021.
PMID: 34055229
Free PMC article.
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Structure-Activity and Brain Kinetics Relationships of 18F-Labeled Benzimidazopyridine Derivatives as Tau PET Tracers.
Watanabe H, Tarumizu Y, Kaide S, Shimizu Y, Iikuni S, Nakamoto Y, Ono M.
Watanabe H, et al. Among authors: tarumizu y.
ACS Med Chem Lett. 2021 Jan 11;12(2):262-266. doi: 10.1021/acsmedchemlett.0c00641. eCollection 2021 Feb 11.
ACS Med Chem Lett. 2021.
PMID: 33603973
Free PMC article.
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